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(4aS,8aR)-1-(4-hydroxybutyl)-6-[2-(3-methylphenyl)acetyl]-decahydro-1,6-naphthyridin-2-one
8-(4-chloro-3-fluorobenzoyl)-2-cyclopropyl-2,8-diazaspiro[5.5]undecan-3-one
1-(2-cyclohexylethyl)-3-hydroxy-3-(1,4-oxazepan-4-ylmethyl)piperidin-2-one
N-benzyl-6-methyl-2-(4-methylphenoxymethyl)-1-[2-(morpholin-4-yl)ethyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
(1R,5R)-6-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-[(2-fluorophenyl)methyl]-N-[(1-hydroxycyclohexyl)methyl]-1,3-benzoxazole-6-carboxamide
N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-(3-chlorophenyl)-N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(2-hydroxyphenyl)propanamide
N-methyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-2,3-dihydro-1,4-benzodioxine-2-carboxamide
5-[(4-hydroxypiperidin-1-yl)methyl]-N-[2-methyl-1-(piperidin-1-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-N-(oxan-4-yl)butanamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{furo[3,2-c]pyridin-4-yl}piperidin-3-ol
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-2,5-dihydro-1H-pyrrole-2-carboxamide
methyl({[2-(3-methylphenyl)pyrimidin-5-yl]methyl}){2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}amine
1-{3-[2-(methoxymethyl)piperidin-1-yl]propyl}-2-methyl-1H-1,3-benzodiazole
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(1H-imidazol-4-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[2-(2-methylpropanesulfonyl)ethyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]propan-1-one
2-(1H-pyrazol-1-yl)-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
2-(4-acetylphenoxy)-N-(quinolin-3-ylmethyl)acetamide
4-(2,4-dioxoimidazolidin-1-yl)-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)benzamide
2-[(2,6-dichlorophenyl)methyl]-5-(4,4-difluoropiperidine-1-carbonyl)pyrimidin-4-ol
3-(azocan-1-yl)-N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]propanamide
(3S,4S)-1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-(4-fluorophenyl)piperidin-3-ol
2-[(3,4-difluorophenyl)methyl]-8-(2-hydroxypropanoyl)-2,8-diazaspiro[4.5]decan-3-one
N-(adamantan-2-yl)-5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carboxamide
6-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1H-indole
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
9-(3-hydroxy-4-methylbenzoyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(3-hydroxyadamantan-1-yl)-N-[1-(2-hydroxyphenyl)ethyl]acetamide
(3S,4R)-1-cyclopentanecarbonyl-4-phenylpyrrolidine-3-carboxylic acid
(1S,5R)-6-(2-methoxyethyl)-3-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
8-(1H-indol-3-ylmethyl)-1-methoxy-1,8-diazaspiro[4.5]decan-2-one
2-(dimethylamino)-2-(4-fluorophenyl)-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]acetamide
5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]pyridin-2-amine
1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
ethyl 2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-1,3-oxazole-4-carboxylate
N-[2-(3-phenylpropoxy)phenyl]oxolane-3-carboxamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(4aS,7aR)-1-[3-(6-oxo-1,6-dihydropyridazin-3-yl)propanoyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-[3-(pyridin-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl]methanol
N-{[6-(dimethylamino)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N-[2-(dimethylamino)ethyl]-3,5-dimethoxybenzamide
N-methyl-N-(2-phenylethyl)-5-({[2-(piperidin-1-yl)ethyl]amino}methyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-({4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
N-(2-methoxyethyl)-1-methyl-N-(naphthalen-1-ylmethyl)azepane-2-carboxamide
ethyl 5-{2-azabicyclo[2.2.1]heptan-2-ylmethyl}-1-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-1H-pyrazole-4-carboxylate
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[(4-phenyloxan-4-yl)methyl]propanamide
2-chloro-4-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidine-1-carbonyl]phenol
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-hydroxyacetamide
N-(1-benzofuran-2-ylmethyl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide