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N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-4-(pyrrolidine-1-sulfonyl)benzamide
1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-4-(morpholin-4-yl)butan-1-one
(2S,4S)-N-ethyl-1-[(5-fluoro-2-methoxyphenyl)methyl]-4-(2-methoxyacetamido)pyrrolidine-2-carboxamide
N-[5-(3-benzyl-1H-1,2,4-triazol-5-yl)-2-methylphenyl]oxolane-2-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-4-(pyridin-3-yl)pyrimidin-2-amine
N-(furan-2-ylmethyl)-2-(1-methylpyrrolidin-3-yl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
(2R,6R)-4-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
5-cyclopropyl-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-N-(thiophen-3-ylmethyl)-1H-pyrazole-4-carboxamide
(3R,4S)-1-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-4-(propan-2-yl)pyrrolidin-3-amine
{1-[(1-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}methanamine
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-4-(dimethylamino)benzamide
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methoxyethyl)piperazine
8-methoxy-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[(2-fluorophenyl)methyl]-4-(4-{[(3S)-2-oxoazepan-3-yl]amino}piperidin-1-yl)benzamide
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-4-(3-methoxybenzoyl)piperazine
5-[(2,3-dimethoxyphenyl)methyl]-8-methoxy-2-[3-(trifluoromethyl)phenyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
8-(butan-2-yl)-1-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
2-methyl-6-{1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperidin-3-yl}pyrimidin-4-ol
(1R,5R)-N,N-dimethyl-6-(4-oxo-1,4-dihydroquinoline-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-methyl-N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}pyrido[2,3-d]pyrimidin-4-amine
6-methoxy-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-{5-[1-(4-chlorophenyl)ethyl]-1,2,4-oxadiazol-3-yl}pyridazine
({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)(quinolin-8-ylmethyl)amine
N-[4-(5-ethylfuran-2-yl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]methanesulfonamide
N-({1-[3-(1,2-oxazinan-2-yl)propanoyl]piperidin-3-yl}methyl)-1-phenylmethanesulfonamide
4-[1-(2-ethoxyethyl)-4-phenyl-1H-imidazol-5-yl]-2-(propan-2-yl)pyrimidine
(4aS,7aR)-1-(2-methyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
({3-[1-(2,4-difluorophenyl)-1H-imidazol-2-yl]phenyl}methyl)dimethylamine
N,N-dimethyl-2-[(1S,5R)-6-{[4-(methylsulfanyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
1-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-3-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]urea
2-(1H-pyrazol-1-yl)-1-[4-(pyrimidin-2-yl)piperazin-1-yl]butan-1-one
8-(3-hydroxy-2-methylbenzoyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-({1-[(3-chloro-4-fluorophenyl)methyl]pyrrolidin-3-yl}methyl)ethane-1-sulfonamide
7-[(4-hydroxy-6-methylquinolin-2-yl)methyl]-N,N,2-trimethyl-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
6-methoxy-3-methyl-N-(5-oxo-1-phenylpyrrolidin-3-yl)-1-benzofuran-2-carboxamide
N-[(2-fluorophenyl)methyl]-3-[1-(4-methylpyrimidine-5-carbonyl)piperidin-3-yl]propanamide
(1-{[3-(cyclopentyloxy)phenyl]methyl}-3-(2-methoxyethyl)piperidin-3-yl)methanol
4-(4-methyl-1H-pyrazol-1-yl)-6-[3-(pentan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyrimidine
2-{1-[(4-methoxypiperidin-1-yl)sulfonyl]azetidin-3-yl}pyridine
2-(dimethylamino)-2-(4-methylphenyl)-1-[4-(thiomorpholin-4-yl)piperidin-1-yl]ethan-1-one
N,N-dimethyl-6-{[(2,3,5-trimethyl-1H-indol-7-yl)methyl]amino}pyridine-3-carboxamide
2-amino-N-[(5-chloro-2-methoxyphenyl)methyl]-N-methyl-4-phenylpyrimidine-5-carboxamide
(4S,4aS,8aS)-1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-4-phenyl-decahydroquinolin-4-ol
N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
methyl 2-({8-cyclopentyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}methyl)-1,3-oxazole-4-carboxylate
(3S,4R)-1-(2,3-dimethylquinoxaline-6-carbonyl)-4-methylpiperidine-3,4-diol
(1R,2R,6S,7S)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
4'-(3-methoxypropyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide