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(5S,9aS,9bS)-5-(4-methoxynaphthalen-1-yl)-2-methyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)pyridine-3-carboxylic acid
1-ethyl-3-(piperidine-1-carbonyl)-N-[2-(propan-2-yloxy)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
(2S,4S)-4-amino-N-methyl-1-[2-(4-methylphenoxy)ethanesulfonyl]pyrrolidine-2-carboxamide
N-{2-[(E)-2-(8-hydroxyquinolin-2-yl)ethenyl]phenyl}-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
methyl N-{[(2S,4S)-4-fluoro-1-[2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetyl]pyrrolidin-2-yl]methyl}carbamate
2-{4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-1,2,3-triazol-1-yl}propanoic acid
2-({4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]phenyl}(methyl)amino)ethan-1-ol
2-ethyl-6-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
1-ethyl-4-[(2-{[(1S,4S)-5-methyl-2,5-diazabicyclo[2.2.1]heptan-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)methyl]-1H-pyrrole-2-carbonitrile
3-(3-methoxypropyl)-1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)piperidine-3-carboxylic acid
1-{2-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]propyl}-1H-indole
2-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-N-methylpyrimidin-4-amine
N-ethyl-3-(3-hydroxy-3-methylbutyl)-N-(pyridin-2-ylmethyl)benzamide
(1S,5R)-6-{[2-(methylsulfanyl)phenyl]methyl}-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-(2-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrimidin-4-yl)piperidin-4-ol
1-(adamantan-2-yl)-4-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
N-benzyl{[6-(phenylamino)pyridin-3-yl]amino}sulfonamide
4-{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}-1,2-dimethylpiperazine
2-[(3R,4S)-3-[1-(methoxymethyl)cyclobutaneamido]-4-(propan-2-yl)pyrrolidin-1-yl]acetic acid
(2S,4S)-4-(2-cyclopentylacetamido)-N-ethyl-1-[(3-hydroxyphenyl)methyl]pyrrolidine-2-carboxamide
N-benzyl-3-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}amino)methyl]-N-methylimidazo[1,2-a]pyridine-2-carboxamide
2-(dimethylamino)-4-methyl-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}pyrimidine-5-carboxamide
(1S,5R)-6-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
1-ethyl-3-(3-methoxyphenyl)-1-(oxan-2-ylmethyl)urea
1-(4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one
3-{[4-(hydroxymethyl)-4-methylpiperidin-1-yl]sulfonyl}-N-(pyrrolidin-3-yl)benzamide
2-(2-ethyl-1H-imidazol-1-yl)-N-[1-methyl-4-(2-oxo-1,3-oxazolidin-3-yl)-1H-indazol-3-yl]acetamide
3-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)-1-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}urea
5-[5-(2-chlorophenyl)furan-2-yl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
3-ethyl-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indole-2-carboxamide
N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)propanamide
2-(2,3-difluorophenoxymethyl)-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]-1,3-oxazole-4-carboxamide
3-benzyl-8-(2,3-dihydro-1H-inden-2-yl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2R,6R)-4-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
8-methoxy-N-methyl-N-(thian-4-yl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1,3-dimethyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl 1-[(3R,5S)-5-(cycloheptylcarbamoyl)-1-(1-ethylpiperidin-4-yl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-benzyl-2-(2,3-difluorophenoxymethyl)-N-ethyl-1,3-oxazole-4-carboxamide
5-{[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-ol
3-[2-(2-methylphenyl)ethyl]-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperidine
1-(1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}azetidin-3-yl)piperidine
5-({[(1-cyclohexylpiperidin-3-yl)methyl](pyridin-3-ylmethyl)amino}methyl)-2-methoxyphenol
6-(2,5-dimethylphenyl)-N-(propan-2-yl)pyridazin-3-amine
4-[(furan-2-ylmethyl)amino]-N-(2-methoxyethyl)-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N,2-diethyl-4-methyl-1,3-oxazole-5-carboxamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N,1,3-trimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)[(4-methylphenyl)methyl]amine
4-{[1-(1-methyl-1H-indole-3-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
(1H-indol-7-ylmethyl)(methyl)[2-(2-methyl-1H-imidazol-1-yl)ethyl]amine