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6-(methoxymethyl)-1-methyl-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-methyl-2-propylpyrimidine
1-(3-phenoxypropyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
butyl 2-(4-methylpiperazin-1-yl)-4-oxo-1,3,8-triazaspiro[4.5]dec-1-ene-8-carboxylate
6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
2-[(1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-3-yl)methyl]-1H-1,3-benzodiazole
ethyl 4-[(4-methoxyphenyl)methyl]-1-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}piperidine-4-carboxylate
2-[benzyl({[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl})amino]ethan-1-ol
4-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-N,N-dimethylpiperazine-1-carboxamide
1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-phenoxyethan-1-one
(3S,4R)-1-(8-chloroquinolin-2-yl)-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
3-(dimethyl-1,2-oxazol-4-yl)-1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]propan-1-one
N-cyclooctyl-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)acetamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)acetamide
3-(azetidine-1-carbonyl)-N-benzyl-N-(cyclopropylmethyl)benzene-1-sulfonamide
2-[(4aS,8aS)-4a-hydroxy-7-(4-methoxypyrimidin-2-yl)-decahydro-2,7-naphthyridin-2-yl]-N,N-dimethylacetamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[3-(4-{[2-(1H-indazol-1-yl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-3-methylbutanamide
2-(2H-1,3-benzodioxole-5-carbonyl)-1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine
N-ethyl-N-(2-hydroxyethyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-{1-[1-(6-cyclopropylpyrimidin-4-yl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
1-(2-{4-[(3-fluorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}-2-oxoethyl)pyrrolidin-2-one
3-[(3R,4S)-1-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
1-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
1-{5-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]thiophen-2-yl}ethan-1-one
N-[3-(1,3-benzothiazol-2-yl)propyl]-4-(1H-pyrazol-3-yl)benzamide
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-2-(1-methyl-3-oxopiperazin-2-yl)acetamide
3-cyclopropyl-N-[1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-1H-pyrazole-5-carboxamide
3-[(3R,4S)-1-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
N,N-dimethyl-5-{1-[2-(1H-pyrazol-4-yl)ethyl]-1H-imidazol-2-yl}pyrimidin-2-amine
4-({4-[3-(pyridin-2-yl)azetidine-1-carbonyl]furan-2-yl}methyl)morpholine
N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]furan-2-carboxamide
[1-(1-{[5-(2-chlorophenyl)furan-2-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methanamine
5-[(2-ethylpyrimidin-4-yl)methyl]-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
4-[(4-fluorophenyl)methyl]-1-(4-methoxypyrimidin-2-yl)-3-(propan-2-yl)-1,4-diazepan-5-one
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(thiophene-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}propan-1-one
butyl 4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxylate
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
2-[(2-methylprop-2-en-1-yl)oxy]-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]benzamide
7-[ethoxy(phenyl)methyl]-4-(quinoxalin-5-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-[2-(3-chloro-4-fluorophenoxy)acetyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
2-{2-[1-(2-methylpyridin-4-yl)-3-phenyl-1H-1,2,4-triazol-5-yl]ethyl}-1,2-oxazinane
(3S,4S)-1-(1-ethyl-1H-pyrazole-4-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
(1-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-[(2-fluorophenyl)methyl]piperidin-3-yl)methanol
{[3-(4-fluorophenyl)oxolan-3-yl]methyl}({[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amine
3-{[1-(4-methylpyridin-2-yl)-3-(phenoxymethyl)-1H-1,2,4-triazol-5-yl]methyl}morpholine
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
11-{[(2-fluorophenyl)methyl]amino}-4-[3-(propan-2-yloxy)propyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(butan-2-yl)[(2-butyl-1H-imidazol-4-yl)methyl](pyridin-4-ylmethyl)amine