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(1S,5R)-3-(2,6-dimethoxypyridine-3-carbonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(1H-imidazol-1-yl)ethyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
2-[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]-5-methylpyrimidin-4-amine
4-[(6-methoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
1-[3-(difluoromethoxy)benzoyl]-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
6-(tert-butylamino)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
(3S,4R)-1-[2-(3-hydroxyphenyl)acetyl]-4-phenylpyrrolidine-3-carboxylic acid
N-(5-cyanopyridin-2-yl)-4-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}benzamide
3-chloro-N-cyclopentyl-4-{[1-(3-hydroxypropanoyl)piperidin-4-yl]oxy}benzamide
N-{[4-methoxy-3-(thiophen-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-{4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-ethoxyethan-1-one
8-methoxy-N-[1-(pyrazin-2-yl)piperidin-4-yl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-({[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}amino)propan-1-ol
N-{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}-3,6-dimethyl-1-benzofuran-2-carboxamide
(2S,4S)-4-[(adamantan-2-yl)amino]-1-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
4-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-3-(3,4,5-trimethoxyphenyl)-1H-pyrazole
1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-4-[2-(pyridin-4-yl)ethyl]piperazine
methyl (2S)-2-[2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamido]-2-phenylacetate
N-methyl-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-(1,2-oxazol-3-ylmethyl)acetamide
6-(hydroxymethyl)-N-{2-[(2-methylprop-2-en-1-yl)oxy]phenyl}-1,4-oxazepane-4-carboxamide
2-methyl-4-(4-{7-methyl-2,7-diazaspiro[4.4]nonane-2-carbonyl}phenyl)butan-2-ol
1-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylpiperidine-1-sulfonamide
7-(3-chlorophenyl)-4-[2-(1H-pyrazol-1-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(1S,5R)-6-(cyclopropylmethyl)-3-[(2-phenylpyrimidin-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(2-methyl-1H-1,3-benzodiazol-5-yl)ethan-1-one
7-methyl-3-[1-(pyridin-3-yl)propan-2-yl]-3H,4H-thieno[3,2-d]pyrimidin-4-one
4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-N-(2-methoxyethyl)-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
1-{7-methylthieno[3,2-d]pyrimidin-4-yl}-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]piperidin-4-amine
8-(2-ethoxyacetyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{2,7-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
4-ethyl-6-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N,N-dimethylpyrimidin-2-amine
4-[4-(1H-1,2,3-benzotriazole-5-carbonyl)piperazin-1-yl]quinazoline
2-ethyl-4-{[3-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}pyrimidine
1-{[(4-fluorophenyl)methyl]carbamoyl}-3-(2-methoxyethyl)piperidine-3-carboxylic acid
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-2-(cyclopropylamino)acetamide
N-[3-(3-methoxyphenyl)phenyl]-1-(pyridine-4-carbonyl)piperidine-2-carboxamide
1-(2-{4-[(4-benzylpiperidin-1-yl)methyl]phenoxy}ethyl)-4-(2,2-dimethyloxane-4-carbonyl)piperazine
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-3-cyclohexyl-1H-pyrazole-4-carboxamide
8-methyl-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
2-amino-6-(2-amino-4-methyl-1,3-thiazol-5-yl)-4-(4-hydroxy-3,5-dimethylphenyl)pyridine-3-carbonitrile
2-{[5-(4-cyclohexyl-1,4-diazepane-1-carbonyl)pyridin-2-yl]amino}ethan-1-ol
6-(4-fluorophenyl)-2-(4-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
3-[3-methyl-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]-N-phenylpropanamide
2-[1-(cyclopropylmethyl)-4-(3,4,7-trimethyl-1H-indole-2-carbonyl)piperazin-2-yl]ethan-1-ol
1-[1-(4-chlorophenyl)ethyl]-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
1-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole