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N-(furan-2-ylmethyl)-2-methanesulfonyl-N-(thiophen-3-ylmethyl)acetamide
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-2-(2,5-dioxoimidazolidin-4-yl)acetamide
2-{2-[(cyclopropylmethyl)sulfanyl]acetyl}-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
methyl (2S,4R)-1-[(3-chloro-4-ethoxyphenyl)methyl]-4-(dimethylamino)pyrrolidine-2-carboxylate
1'-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-(2,5-difluorophenyl)-4-[4-(2-hydroxyethyl)piperazin-1-yl]piperidine-1-carboxamide
5-ethyl-N4-methyl-N4-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]pyrimidine-2,4-diamine
N-(1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperidin-4-yl)methanesulfonamide
methyl 5-{7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-5-oxopentanoate
3-(2-methyl-5-oxopyrrolidin-2-yl)-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]propanamide
3-(2-chlorophenyl)-N,5-dimethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1,2-oxazole-4-carboxamide
5-[({2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}carbamoyl)amino]-2-methoxy-N,N-dimethylbenzamide
N,N-dimethyl-9-oxo-8-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecane-2-sulfonamide
1-(1-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)propan-1-ol
4-(4-propylbenzoyl)-1λ6-thiomorpholine-1,1-dione
2-(3-methoxypropyl)-9-(trimethyl-1H-pyrazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
3-methyl-4-{1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}-1,2,5-oxadiazole
9-(3-ethyl-1,2-oxazole-5-carbonyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-amino-N-methyl-4-phenyl-N-(thiophen-3-ylmethyl)-1H-pyrazole-3-carboxamide
1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-2-[2-(trifluoromethyl)phenyl]ethan-1-one
2-(pyridin-2-ylmethyl)-9-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
(2E)-3-(2-chlorophenyl)-1-[9-(oxan-2-ylmethoxy)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]prop-2-en-1-one
1-{1-[(3-chloro-4-fluorophenyl)methyl]azetidin-3-yl}piperidine
(1S,5R)-6-(2,5-dimethylfuran-3-carbonyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-{1-[(dimethyl-1,3-thiazol-5-yl)methyl]-1H-imidazol-2-yl}pyridine
(4aS,8aR)-6-[2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetyl]-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(4-methylphenyl)piperazine
N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-6-(pyrimidin-5-yl)pyridine-3-carboxamide
1-[3-(2-fluorophenyl)pyrrolidin-1-yl]-3-(3-hydroxy-1,2-oxazol-5-yl)propan-1-one
N-{[(3S,4S)-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3-hydroxypiperidin-4-yl]methyl}pyrrolidine-1-carboxamide
N-(3-{[(4-fluorophenyl)methyl]sulfanyl}propyl)-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N,1-dimethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-phenyl-3-[1-(1H-1,2,3-triazole-5-carbonyl)piperidin-4-yl]-1H-indole
1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-4-(thiophen-2-ylmethyl)-1,4-diazepane
(furan-2-ylmethyl)[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl](pyridin-2-ylmethyl)amine
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-5-methylpiperidin-2-one
3-(4-methoxyphenyl)-3-phenyl-1-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}propan-1-one
2-{2-[1-(3-fluorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
7-[(2,3-difluorophenyl)methyl]-2-(5-methyl-1,3-oxazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(4,5,6,7-tetrahydro-1-benzothiophen-3-yl)ethyl]-1H-1,2,3-triazole-5-carboxamide
3-[(3R,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-fluorophenyl)urea
N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-[(2,5-dimethoxyphenyl)methyl]-N'-(3,5-dimethylphenyl)propanediamide
1-[(1-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}pyrrolidin-2-yl)methyl]-1H-pyrazole
5-{[8-(3-hydroxypropyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
1-[(4aR,8aS)-6-(3-phenoxypropanoyl)-decahydro-1,6-naphthyridin-1-yl]-4-methylpentan-1-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-5-phenyl-1,2-oxazole-3-carboxamide
N-methyl-N-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
4-phenyl-3-{[1-(pyridin-3-ylmethyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(4aS,8aR)-4a-(hydroxymethyl)-6-(pyridine-4-carbonyl)-decahydro-1,6-naphthyridin-1-yl]-2-(methylsulfanyl)ethan-1-one