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methyl 4-({2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamido}methyl)benzoate
1-[1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-4-yl]-3-phenylpropan-1-ol
4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-1-(4-methylphenyl)piperidine
N-(2-methoxyethyl)-1-[1-(1,3-thiazol-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]acetamide
(1S,5R)-6-(2-methoxyethyl)-3-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}benzamide
1-[(3-chloro-4,5-dimethoxyphenyl)methyl]-2-(5-methyl-1,2-oxazol-3-yl)piperidine
(3S,5R)-N3-butyl-N5-(2,3-dihydro-1H-inden-5-yl)piperidine-3,5-dicarboxamide
2-{6-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-methylpyrimidin-4-yl}ethan-1-amine
6,7-dimethoxy-2-{1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}-1,2,3,4-tetrahydroisoquinoline
1-(3,5-dimethyl-4-{2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-1H-pyrrol-2-yl)ethan-1-one
1-benzyl-5-(4-benzylpiperidine-1-carbonyl)-4-oxo-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
1-[(2-fluorophenyl)methyl]-N-[(3-phenylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(azepan-1-yl)-2-phenylethyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-[2-(4-fluorophenyl)morpholin-4-yl]-1,3-dimethyl-1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid
2-{[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}-2-(3-methoxyphenyl)acetic acid
[(3-{[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(thiophen-2-ylmethyl)amine
6-[(2E)-3-(4-fluorophenyl)prop-2-enoyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
(3R,4R)-1-{[4-ethoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
2-{1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]pyrrolidin-3-yl}benzoic acid
2-(2-ethyl-1H-imidazol-1-yl)-1-[2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]ethan-1-one
2-cyclopentyl-9-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
(1R,3S)-3-[4-(benzyloxy)-4-(prop-2-en-1-yl)piperidine-1-carbonyl]cyclopentan-1-amine
N-(1-{7-[(4-methoxy-2,3-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
methyl 2-(diethylsulfamoyl)-6-[2-(2,3-difluorophenyl)acetyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-{[(3-fluorophenyl)methyl]amino}-N,5-dimethyl-N-(2-methylpropyl)thieno[2,3-d]pyrimidine-6-carboxamide
N4-cyclopropyl-6-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrimidine-2,4-diamine
2-(5-methyl-1H-pyrazol-1-yl)-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
4-(3-acetylbenzoyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
5-chloro-N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-2,3-dihydro-1H-indole-2-carboxamide
2-(1-{[2-(5-methylfuran-2-yl)phenyl]methyl}pyrrolidin-2-yl)ethan-1-ol
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(3-methylphenyl)methyl]piperidine
(3S,9R)-11-(3,5-dichlorobenzoyl)-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
5-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]-2-(pyridin-4-yl)pyrimidin-4-ol
1-(8-chloro-2-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-4-(thiophen-2-yl)butan-1-one
2-methoxyethyl 2-[(3-methoxyphenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decane-8-carboxylate
3-{5-[(1-methyl-1H-imidazol-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-(4-methylpiperazin-1-yl)propan-1-one
4-({2-[(2-chloro-6-fluorophenyl)methoxy]phenyl}methyl)piperazin-2-one
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
(3R,4S)-1-cyclopentanecarbonyl-4-(3-methoxyphenyl)pyrrolidin-3-amine
6-[2-(oxan-2-yl)ethyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[2-(2-phenylethyl)morpholin-4-yl]propan-1-one
1-{3,5-dimethyl-4-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-1H-pyrrol-2-yl}ethan-1-one
[(1S,3S,3aS,6aR)-5-methyl-3-(6-methyl-2H-1,3-benzodioxol-5-yl)-1-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
N-(1,1-dioxo-1λ6-thian-4-yl)-8-fluoro-N-methylquinoline-2-carboxamide
8-[2-(dimethylamino)acetyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl 3-({3-cyclohexyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)benzoate
7-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one