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1-(difluoromethyl)-4-[3-(1-methoxyethyl)phenyl]-5-methyl-1H-pyrazole
(2R)-N-[1-benzyl-6-(propan-2-yloxy)-1H-indazol-3-yl]-5-oxopyrrolidine-2-carboxamide
1-methyl-5-{3-[3-(4-methylpiperazin-1-yl)-3-oxopropyl]piperidine-1-carbonyl}-1H-pyrrole-3-carbonitrile
1-[2-(2,3-dimethoxyphenyl)ethyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
N-[(2R,3R)-2-ethoxy-1'-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
(3aS,6aS)-2-(1,3-benzoxazol-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-6-methoxy-1-methyl-1H-indole-2-carboxamide
2,2-dimethyl-4-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
N-{2-[cyclopentyl(methyl)amino]ethyl}-N-methyl-6-(propan-2-yl)pyrimidin-4-amine
N-[2-(4-methoxybenzenesulfonamido)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-(cyclohexylmethyl)-N-[3-(dimethylamino)-2,2-dimethylpropyl]-1H-1,2,3-triazole-4-carboxamide
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]acetamide
2-methyl-6-{5-[2-(pyrazin-2-yl)ethyl]-1H-1,2,4-triazol-1-yl}-1,3-benzothiazole
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carboxamide
5-methoxy-1-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-indole-2-carboxamide
[(3-ethoxy-4-methoxyphenyl)methyl][(1-methylpiperidin-3-yl)methyl](2-phenylethyl)amine
8-hydroxy-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]quinoline-7-carboxamide
2-benzyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,3-benzoxazole-5-carboxamide
2-{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1,2-oxazinane
N-[(2,4-dimethylphenyl)(pyridin-3-yl)methyl]-2-ethylpyrimidine-5-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-3-(5-ethylthiophene-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[1-(5-chloropyridin-2-yl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
4-(hydroxymethyl)-1-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperidin-4-ol
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-(3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)acetamide
3-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-1-[2-methoxy-5-(4H-1,2,4-triazol-4-yl)phenyl]urea
4-cyclopentyl-N-[3-methyl-1-(propan-2-yl)-1H-pyrazol-5-yl]-3-oxopiperazine-1-carboxamide
1-(1,5-dimethyl-1H-pyrrole-2-carbonyl)-3-phenylpiperazine
1-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-oxo-N-(propan-2-yl)-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
(1S,5R)-3-[2-(methylsulfanyl)acetyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(4-phenylpiperidin-1-yl)-N-[1-(pyrazin-2-yl)propan-2-yl]acetamide
6-(1-{4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}piperidin-4-yl)-2-methylpyrimidin-4-ol
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-4-(1H-imidazol-1-yl)butanamide
3-({[1-(2-chloroprop-2-en-1-yl)-7-(methylsulfanyl)-2-oxo-1,2-dihydroquinolin-3-yl]methyl}amino)-1λ6-thiolane-1,1-dione
ethyl 4-[({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)amino]piperidine-1-carboxylate
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-(3-{[ethyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)amino]methyl}phenyl)ethan-1-one
2-methoxy-N-[2-(1H-pyrrole-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
1-(5-fluoro-1H-indole-2-carbonyl)-N-(4-fluorophenyl)piperidin-3-amine
1-benzyl-N3-(2,3-dihydro-1H-inden-2-yl)-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
6-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-2-carbonitrile
(3aR,5R,6S,7aS)-2-(4-amino-5-methylpyrimidin-2-yl)-octahydro-1H-isoindole-5,6-diol
2-(4-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-(3-methylbut-2-en-1-yl)piperazin-2-yl)ethan-1-ol
4-(4-methylphenoxy)-1-(1-methylpiperidine-2-carbonyl)piperidine
1-(5-chloro-2-hydroxybenzoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazole
(4aR,8aR)-2-[(1-propyl-1H-imidazol-2-yl)methyl]-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
1-ethyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydropyridin-2-one
3-[(3R,4S)-4-(morpholin-4-yl)-1-[4-(trifluoromethyl)benzoyl]piperidin-3-yl]propan-1-ol
1-cyclopropyl-4-[({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]pyrrolidin-2-one