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4-(7-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}pyrazolo[1,5-a]pyrimidin-5-yl)pyridine
5-methyl-N-[2-(propylsulfanyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
(2E)-N-({3-methyl-7-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinane-4-carbonyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-phenylprop-2-enamide
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
8-(5-chlorothiophene-2-carbonyl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
N-propyl-5-[4-(1H-pyrazol-1-yl)phenyl]furan-2-carboxamide
N-tert-butyl-2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-cycloheptyl-3-(2-hydroxyphenyl)-3-(4-hydroxyphenyl)propanamide
(1R,5R)-N,N-dimethyl-6-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-(3-{2-amino-3-cyano-5H,7H,8H-pyrano[4,3-b]pyridin-4-yl}-1H-indol-1-yl)acetic acid
4-benzyl-3-[1-(2-propoxyacetyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-ethyl-1-methyl-3-({1-[3-(1,2-oxazinan-2-yl)propanoyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{2-chloro-4-[2-(2-methoxyphenyl)acetamido]phenyl}propanamide
1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-4-(methoxymethyl)piperidine
N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-2-(3-phenylpyrrolidin-1-yl)acetamide
1-[(3,5-dimethylphenyl)methyl]-4-[4-(hydroxymethyl)-1,3-thiazol-2-yl]piperazin-2-one
N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
2-(2-methoxyphenyl)-N-(1-{2-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)acetamide
5-amino-4-chloro-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-1H-pyrazole-3-carboxamide
3-benzyl-5-(but-3-en-1-yl)-1H-1,2,4-triazole
1-[1-(2-cyclohexylacetyl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
2-(cyclopropylmethyl)-8-[2-(4-ethylphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
2-cyclobutyl-1-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-4-yl)-5-fluoro-1H-1,3-benzodiazole
(2S)-1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxamide
9-(1-methyl-1H-pyrazole-5-carbonyl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-cyclohexyl-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}pyrimidine
(2E)-3-(2-chlorophenyl)-1-{4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}prop-2-en-1-one
3-(3-methoxypropyl)-1-[2-(thiophen-3-yl)acetyl]piperidine-3-carboxylic acid
N-[(1-methylpyrrolidin-3-yl)methyl]-5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-amine
(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)[(3-phenyl-1H-pyrazol-4-yl)methyl]amine
4-[2-(4-methyl-1,4-diazepane-1-carbonyl)-1-benzofuran-5-yl]-1-(3-phenylbutyl)piperidin-4-ol
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-2-oxo-4-phenylbutanamide
(2R,6R)-4-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-{[3-({1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}oxy)phenyl]methyl}-4-(pyridin-3-ylmethyl)piperazine
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]propanamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(2-methylprop-2-en-1-yl)-1,3-oxazole-4-carboxamide
N-{[3-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-5-methyl-N-(pyridin-2-ylmethyl)thiophene-2-carboxamide
1-[(4aR,8aR)-7-{[6-(dimethylamino)pyridin-3-yl]methyl}-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
1-{4-[({5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)methyl]piperidin-1-yl}ethan-1-one
5-[(4-hydroxyphenyl)methyl]-1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-methyl-4-[5-methyl-3-(pyridin-2-yl)-1H-1,2,4-triazol-1-yl]pyridine
N-benzyl-N-methyl-3-[1-(quinolin-2-yl)piperidin-4-yl]propanamide
N-ethyl-5-[4-(quinazolin-4-yl)piperazine-1-carbonyl]pyrimidin-2-amine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
2-(2,5-dioxoimidazolidin-1-yl)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
N-benzyl-1-methyl-5-(1,2,3,4-tetrahydronaphthalen-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)cyclobutanecarboxamide
2-(2-{methyl[2-(1H-pyrazol-4-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
5-{4-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one