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4-(ethanesulfonyl)-2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)phenol
methyl 1-[2-(1H-indol-3-yl)ethyl]-3-(3-methoxypropanamido)-5-[(quinolin-8-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-(2,3-dihydro-1H-inden-2-yl)-11-{[2-(pyridin-3-yl)ethyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N5-benzyl-N6-[(3-methyloxetan-3-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
4-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-N,N-dimethylaniline
3-[(4aS,8aS)-decahydroisoquinolin-2-yl]-N-(2-methylphenyl)-3-oxopropanamide
2-({[(3R,4R)-1-[1-(4-chlorophenyl)cyclobutanecarbonyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
5-ethyl-2-{1-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}pyridine
N-methyl-5-({2-[2-(thiophen-2-yl)ethyl]piperidin-1-yl}methyl)furan-2-carboxamide
2-(adamantan-1-yl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}acetamide
(1R,5S,6S)-6-[3-(3-methylphenoxy)azetidine-1-carbonyl]-3-azabicyclo[3.1.0]hexane
(4aS,7aR)-1-(1-methyl-1H-pyrrole-2-carbonyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{5-[2-(methylsulfanyl)pyridin-3-yl]-1H-1,2,4-triazol-1-yl}butan-2-ol
4-{[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]carbonyl}imidazolidin-2-one
methyl 2-[1-(2,3-dihydro-1H-inden-5-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]acetate
4-[2-(methylsulfanyl)ethyl]-2-oxo-7-(pyrrolidin-1-yl)-1,2,3,4-tetrahydroquinoline-6-carboxamide
N-methyl-1-(1-methylpiperidin-4-yl)-N-(pyrazin-2-ylmethyl)piperidine-3-carboxamide
3,5-dimethyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)-1-benzofuran-2-carboxamide
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[(1-phenylcyclopentyl)methyl]propanamide
2-[4-phenyl-1-(pyridin-3-ylmethyl)-1H-imidazol-5-yl]benzoic acid
2-methyl-1-{[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}-4-(4-methylphenyl)piperazine
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-2-(4-methoxyphenyl)acetamide
(3R,4R)-4-cyclobutyl-1-[1-(3-methoxyphenyl)piperidin-4-yl]-3-methylpiperidin-4-ol
N-butyl-5-(2,6-difluorophenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
2-[(isoquinolin-5-yloxy)methyl]-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1,3-oxazole-4-carboxamide
(2S,4S)-N-ethyl-1-(naphthalen-1-ylmethyl)-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
2-(dimethylamino)-2-(2-methylphenyl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
1-[(3-methoxyphenyl)methyl]-5-methyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
N-[2-(3,5-dimethylphenoxy)ethyl]-3-fluoro-N,5-dimethylimidazo[1,2-a]pyridine-2-carboxamide
N,N-dipropyl-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
4-chloro-N,N-diethyl-3-[2-(2-hydroxyphenoxy)acetamido]benzamide
5-[4-(3-methoxybenzoyl)piperazine-1-carbonyl]-2-(methylsulfanyl)pyrimidine
3-(azetidine-1-sulfonyl)-N-(1,4-dioxan-2-ylmethyl)-N-methylbenzamide
N-[2-(1-methylpiperidin-3-yl)ethyl]-2-(propan-2-ylsulfanyl)acetamide
N-[2-(5-methylfuran-2-yl)ethyl]-3-{[(2R)-oxolan-2-ylmethyl]sulfamoyl}benzamide
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl 2-({3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecan-8-yl}methyl)-1,3-oxazole-4-carboxylate
[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]({[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl})amine
5-{[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]methyl}-N-methyl-1,2,4-oxadiazole-3-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-1-{1-oxa-8-azaspiro[4.5]decan-8-yl}ethan-1-one
3-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-N-[2-(1,3-thiazol-2-yl)ethyl]benzene-1-sulfonamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(piperidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(4-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-cyclohexylpiperazin-2-yl)ethan-1-ol
(3S,4R)-1-ethyl-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
1-[(2-ethylpyrimidin-5-yl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
N-[1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
2-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}pyridine-4-carbonitrile
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-[2-(furan-2-yl)ethyl]acetamide
N-{2-[2-(2,4-dioxoimidazolidin-1-yl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}oxolane-2-carboxamide
6-(cyclopentylamino)-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]pyridine-3-carboxamide