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2-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-6-methoxypyrimidin-4-amine
2-(4-ethylpiperazin-1-yl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
(2S)-2-amino-3-(1H-imidazol-4-yl)-1-[4-(4-methoxybenzoyl)piperazin-1-yl]propan-1-one
4-(1-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1H-imidazol-2-yl)pyridine
4-{4-[(2-methyl-1,3-oxazol-4-yl)methyl]-2-oxopiperazin-1-yl}benzonitrile
4-{2-[(2-methoxyethyl)(methyl)amino]acetyl}-1-(2-methylphenyl)piperazin-2-one
(3R,4S)-4-phenyl-1-{[5-(1H-pyrazol-5-yl)furan-2-yl]sulfonyl}pyrrolidin-3-amine
1-[(3S,4R)-1-({9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
2-{[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}benzoic acid
2-{3-[2-amino-3-cyano-6-(4-methoxyphenyl)pyridin-4-yl]phenoxy}acetamide
5-(oxolan-3-ylmethyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-(2-methylpropyl)-1-[1-(2-phenoxyacetyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
1-butyl-3-[2-(2,2-dimethyl-3-oxopiperazin-1-yl)-2-oxoethyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
2-cyclobutanecarbonyl-N-(5-methyl-1,3,4-thiadiazol-2-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
3-[1-(3,6-dimethylpyrazin-2-yl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(4aS,8aR)-1-butyl-6-(3,3,3-trifluoropropyl)-decahydro-1,6-naphthyridin-2-one
2-chloro-5-acetamido-N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]benzamide
3-{2-[2-(4-hydroxyphenyl)ethyl]piperidine-1-carbonyl}-1,6-dimethyl-1,2-dihydropyridin-2-one
2-cyclopentyl-1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]ethan-1-one
6-tert-butyl-2-[4-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
N-{[2-(azepan-1-yl)-7-methylquinolin-3-yl]methyl}-N-(3-methoxypropyl)-2-methylpropanamide
1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
3-(4-methyl-1,3-thiazol-5-yl)-N-[(4-methylphenyl)(pyridin-4-yl)methyl]propanamide
(1S,5R)-6-(cyclobutylmethyl)-3-(6-oxo-1,6-dihydropyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-chlorophenyl)urea
(2S,4S)-4-amino-1-(3,4-dimethylbenzoyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-(1-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1H-imidazol-2-yl)benzonitrile
N,N-diethyl-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(1S,4S)-2-({2-[3-(4-methylpiperazin-1-yl)propoxy]phenyl}methyl)-2-azabicyclo[2.2.1]heptane
2-[4-(1-methyl-1H-pyrazol-4-yl)-1H-pyrazol-1-yl]-N-{1-[(5-methylfuran-2-yl)methyl]-1H-pyrazol-5-yl}acetamide
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-{[(4-methoxy-2,5-dimethylphenyl)methyl]amino}pyrrolidine-2-carboxamide
(2S)-N-ethyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-1-(piperidin-4-yl)pyrrolidine-2-carboxamide
(3S)-N-tert-butyl-2-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
(1-{4-[4-({[1-(morpholin-4-yl)cyclopentyl]methyl}amino)piperidin-1-yl]benzoyl}piperidin-3-yl)methanol
1-[(4aR,8aR)-4a-hydroxy-7-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
3-{[2-(3-phenyl-1,2-oxazol-5-yl)-1H-imidazol-1-yl]methyl}-1λ6-thiolane-1,1-dione
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-1-methylpiperidine-2-carboxamide
3-(1-methylpiperidin-2-yl)-N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}propanamide
N-cyclopropyl-2,3-dimethyl-N-{[3-(2-methylpropoxy)phenyl]methyl}-1H-indole-7-carboxamide
N-[(1S,2R)-2-aminocyclobutyl]-1,3,5-trimethyl-1H-pyrazole-4-sulfonamide
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-N-methyl-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-cyclopentyl-4-(1H-imidazol-2-ylmethyl)piperazin-2-one
2-[(4-{4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-yl}piperidin-1-yl)methyl]phenol
3-(3-chloro-1,2-oxazol-5-yl)-1-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propan-1-one
naphthalen-1-yl (7R,9aR)-7-benzyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
methyl 6-benzoyl-2-{[(2-fluorophenyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-{[(5-methyl-1H-pyrazol-3-yl)methyl]sulfamoyl}-N-(pyridin-3-yl)benzamide
6-methoxy-3-{[(2S)-4-methyl-2-phenylpiperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[(3-methylphenyl)methyl](propan-2-yl)amine