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1-{imidazo[1,2-a]pyridine-3-carbonyl}-3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine
5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-N-(2,2,2-trifluoroethyl)-1H-pyrazole-3-carboxamide
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
2-(dimethylamino)-N-methyl-2-(2-methylphenyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
[(1-cyclopentylpiperidin-4-yl)methyl](pyridin-3-ylmethyl)(quinolin-4-ylmethyl)amine
4-{[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]methyl}-5-(hydroxymethyl)-2-methylpyridin-3-ol
5-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrazin-2-amine
4-benzyl-3-[1-(3-methyl-1,2-oxazole-5-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(4-phenylpiperazin-1-yl)-3-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]propan-1-one
2-(2,5-dioxoimidazolidin-1-yl)-N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}acetamide
N-[2-methyl-5-(2-oxopyrrolidin-1-yl)phenyl]-3-propylmorpholine-4-carboxamide
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(1S,5R)-3-benzyl-6-(2-methyl-1,3-thiazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
2,3,6-trifluoro-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)benzamide
2-[5-({4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}methyl)-1,2,4-oxadiazol-3-yl]pyrazine
2-benzyl-N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-1,3-thiazole-4-carboxamide
1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperidin-4-amine
N-(2-methoxyethyl)-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
(1R,3S)-3-amino-N-[(4-fluorophenyl)methyl]-N-[(2-methoxyphenyl)methyl]cyclohexane-1-carboxamide
8-{[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-3-azaspiro[5.5]undecan-9-amine
N-cyclopropyl-1-{1-[4-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl}piperidine-3-carboxamide
4-{1-[5-(2-chlorophenyl)furan-2-carbonyl]piperidin-3-yl}morpholine
5-(3,4-dimethoxyphenyl)-1,2,3,4-tetrahydroisoquinoline
[(3R,4R)-4-[(dimethylamino)methyl]-1-{thieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl]methanol
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-3-(3-methoxyphenyl)propanamide
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
(3S)-1-({3-methoxy-4-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)pyrrolidin-3-amine
4-hydroxy-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
(4S)-3-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-4-(propan-2-yl)-1,3-oxazolidin-2-one
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(pyrimidin-2-yl)piperidin-4-amine
5-cyclopropanecarbonyl-1'-[(1-propyl-1H-imidazol-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
6-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(3-chlorophenyl)-4-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazine
3-{1-[2-(2-oxo-4-phenylpyrrolidin-1-yl)acetyl]piperidin-4-yl}benzonitrile
1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-phenylpiperidine
1-(cyclohexylmethyl)-3-hydroxy-3-({[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}methyl)piperidin-2-one
1-methyl-3-(propan-2-yl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(prop-2-en-1-yl)(pyridin-3-ylmethyl)(quinolin-4-ylmethyl)amine
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amine
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(2,2,2-trifluoroethyl)piperidine-3-carboxamide
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-1-[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]propan-1-one
(4aS,7aR)-1-(1-aminocyclopropanecarbonyl)-4-[(3,5-dimethylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-(1-benzothiophene-2-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-(4-{[2-(2-phenylethynyl)phenyl]methyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[5-methyl-2-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}urea
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-6-(pyrrolidine-1-carbonyl)pyrazin-2-amine
1-[(2-methoxyphenyl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid