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4-methoxy-N-({1-[(5-methylthiophen-2-yl)methyl]piperidin-3-yl}methyl)benzene-1-sulfonamide
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-1,2-oxazole-3-carboxamide
3-butyl-1-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}phenyl)urea
3-{[(2,3-dihydro-1H-inden-2-yl)amino]methyl}-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
5-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-2-(pyridin-2-yl)pyrimidine
[(1R,3R,3aS,6aR)-5-benzyl-3-[1-(propan-2-yl)piperidin-4-yl]-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
4-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyridine
2-(3-methylbutyl)-8-[(3-methylpyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
5-[(1R,5S)-6-azabicyclo[3.2.1]octane-6-carbonyl]-2-(3-phenylpropyl)-1,3-benzoxazole
4-(furan-3-yl)-6-methyl-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
[4-(1-benzothiophen-2-yl)pyridin-2-yl]methanol
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-2-(2H-indazol-2-yl)acetamide
2-[2-benzyl-4-(3-methoxyphenyl)-5-oxopiperazin-1-yl]-N-methylacetamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[2-(dimethylamino)-6-methylpyrimidin-4-yl]piperazin-2-one
(4aR,7aS)-1-(1H-imidazol-2-ylmethyl)-4-(quinolin-5-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3aS,6aS)-2-(4-acetylbenzoyl)-5-cyclopentyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[(5-methylpyrazin-2-yl)methyl]-9-[(5-propylfuran-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-3-[(5-chloro-3-methyl-1H-indol-2-yl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
2-{3,5-dimethyl-4-[2-(pyridin-4-ylsulfanyl)acetamido]-1H-pyrazol-1-yl}acetic acid
3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]propanamide
N-[(1R)-2,3-dihydro-1H-inden-1-yl]-2-(dimethylamino)-4-methylpyrimidine-5-carboxamide
3-(2-chlorophenyl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-phenylpropanamide
1-(2-{1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-2-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
[(3R,4R)-1-(3-chloro-5-fluorobenzoyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
(4aR,7aS)-1-[2-(dimethylamino)acetyl]-4-(pyrrolidine-1-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]acetamide
N-[3-(1H-imidazol-1-yl)propyl]-3-phenyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]-2-methyl-1H-pyrrole-3-carboxamide
N-methyl-N-[(3-methylpyridin-4-yl)methyl]-2-(pyridin-2-yl)acetamide
3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(2-oxo-1,2-dihydropyridin-1-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)propanamide
2-[4-(2-chloro-4-fluorophenyl)-1H-pyrazol-1-yl]-N-methylacetamide
7-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-2-oxa-7-azaspiro[4.5]decan-8-one
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzamide
(1S,5R)-6-(cyclobutylmethyl)-3-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
7-(2-hydroxyethyl)-2-[3-(4H-1,2,4-triazol-4-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
(5S,9aS,9bS)-2-[(4-methoxyphenyl)methyl]-5-(1-methyl-1H-indol-3-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N'-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-N-(propan-2-yl)ethanediamide
2-[methyl({5-[2-(methylsulfanyl)pyridine-3-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]ethan-1-ol
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamide
N-(1-benzoylpiperidin-4-yl)-2-(2,3-dihydro-1H-inden-1-yl)acetamide
(2-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}-1,3-thiazol-4-yl)methanol
N-[(3R,4S)-4-cyclopropyl-1-[2-(4-fluorophenoxy)ethyl]pyrrolidin-3-yl]-3-hydroxypropanamide
N-(3-ethoxypropyl)-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(1H-pyrazol-1-yl)acetamide
4-(4-{1-[4-(pyrrolidin-1-yl)butyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
1-(4-methylpiperazin-1-yl)-3-{1-[2-(methylsulfanyl)benzoyl]piperidin-3-yl}propan-1-one
1-[(2-chlorophenyl)methyl]-4-(thiophen-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-{1'-[(2-fluorophenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one