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N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
N,N-dimethyl-5-[4-(2-methylpyrrolidine-1-carbonyl)quinolin-2-yl]pyrimidin-2-amine
N-[1-(4-chlorophenyl)ethyl]-N-methyl-4-(1H-pyrazol-4-yl)butanamide
ethyl 3-{2-[(2-ethoxyphenyl)carbamoyl]acetamido}hexanoate
(3S,4R)-1-[(2-cyclohexylpyrimidin-5-yl)methyl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-ethylpyrimidine-5-carboxamide
2-{[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-4,5,6,7-tetrahydro-1,3-benzothiazole
(2E)-1-{3-[5-(2-fluorophenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}-3-(thiophen-2-yl)prop-2-en-1-one
1-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)but-2-yn-1-one
(4aR,7aS)-1-(2-hydroxyethyl)-4-[(3-methoxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-benzenesulfonamido-1-ethyl-N-[(4-fluorophenyl)methyl]-N,2-dimethyl-1H-1,3-benzodiazole-7-carboxamide
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]ethan-1-one
8-(3-methanesulfonylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-amino-6-(furan-2-yl)-4-(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)pyridine-3-carbonitrile
6-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-5,6,7,8-tetrahydro-1,6-naphthyridine
1-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
(1S,4S)-2-(2-methoxy-5-phenylphenyl)-5-(1-methylcyclopropanecarbonyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}benzamide
ethyl 2-[(4-acetyl-4-phenylpiperidine-1-carbonyl)amino]-1H-imidazole-5-carboxylate
1-(azepan-1-yl)-2-{4-[2-(methylsulfanyl)pyridine-3-carbonyl]morpholin-3-yl}ethan-1-one
2-(3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}pyrrolidin-1-yl)-N-(propan-2-yl)acetamide
N-methyl-1-[3-(methylsulfanyl)propyl]-N-(2-phenylethyl)piperidin-3-amine
1-ethyl-4-({2-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}methyl)pyrrolidin-2-one
1-(1-benzylpiperidin-4-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine-3-carboxamide
5-{[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]carbamoyl}thiophene-2-carboxylic acid
2-[(1S,5R)-3-[2-(3,5-difluorophenyl)acetyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]quinoxaline-5-carboxamide
2-[(3-methylphenyl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
(3aR,6aR)-2-[(2,3-dimethoxyphenyl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{3-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]-1H-pyrazol-1-yl}-N-(1-methyl-1H-pyrazol-5-yl)acetamide
6-[1-(3-methylphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
2-benzyl-8-(1-methyl-2-oxoimidazolidine-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
N2,N4,N4,5-tetramethyl-N2-(1,2-oxazol-5-ylmethyl)pyrimidine-2,4-diamine
2-(1,3-thiazol-2-yl)-N-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]piperidine-1-carboxamide
N,N,4,5-tetramethyl-6-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]pyrimidin-2-amine
2-[6-hydroxy-4-(pyrazin-2-yl)-1,4-diazepan-1-yl]-1-(piperidin-1-yl)ethan-1-one
4-[1-(2-methanesulfonylethyl)-4-phenyl-1H-imidazol-5-yl]-2-(propan-2-yl)pyrimidine
(3aR,6aS)-5-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-methyl-5-{5-[4-(piperidin-1-ylmethyl)phenyl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
2-[1-(3-butanamidobenzoyl)-3-oxopiperazin-2-yl]acetic acid
3-({2-cyclopropyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}(methyl)amino)-1-phenylpropan-1-ol
methyl(naphthalen-1-ylmethyl)[(3-{2-[4-(thiophene-2-sulfonyl)piperazin-1-yl]ethoxy}phenyl)methyl]amine
1-benzyl-N,N-dimethyl-5-{[(3-methylphenyl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N2-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-5-fluoro-N4,N4-dimethylpyrimidine-2,4-diamine
N-[(5-methylpyrazin-2-yl)methyl]-4-(piperidin-1-ylmethyl)benzamide
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2-methylimidazo[1,2-a]pyridine-6-carboxamide
3-hydroxy-5-[4-(1H-pyrazol-5-yl)phenyl]benzoic acid
3-oxo-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-1,2,3,4-tetrahydroquinoxaline-6-carboxamide