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(3R,4R)-1-[(3-chloro-2-fluorophenyl)methyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-(2-methoxyethyl)-N-methylpyrimidine-5-carboxamide
({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)[2-(oxan-4-yl)ethyl]amine
3-methyl-1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}but-2-en-1-one
2-chloro-3-{[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}-9-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
2-methyl-4-(2-methylphenyl)-1-{pyrazolo[1,5-a]pyridine-7-carbonyl}piperazine
3-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-1-[2-fluoro-5-(4H-1,2,4-triazol-4-yl)phenyl]urea
3,6,7-trimethyl-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-1-benzofuran-2-carboxamide
N-methyl-N-[1-({4-[6-oxo-4-(pyridin-3-yl)-1,6-dihydropyrimidin-2-yl]phenyl}methyl)pyrrolidin-3-yl]acetamide
(3S,4R)-4-(pyridin-4-yl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}pyrrolidine-3-carboxylic acid
2-[5-(3-benzoylpiperidine-1-carbonyl)-1H-1,3-benzodiazol-1-yl]ethan-1-ol
4-(5-methylpyridin-2-yl)-1-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperidin-4-ol
(3S,4S)-1-[3-methyl-4-(1H-pyrrol-1-yl)benzoyl]piperidine-3,4-diol
6-chloro-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}imidazo[1,2-a]pyrimidine-2-carboxamide
methyl 1-methyl-5-({[2-(2-methylphenoxy)pyridin-3-yl]methyl}carbamoyl)-1H-pyrazole-3-carboxylate
1-{5-[3-(3-methylbutanoyl)piperidine-1-carbonyl]pyridin-2-yl}piperidine-4-carboxamide
N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]pyrazolo[1,5-a]pyridine-3-carboxamide
2-methyl-8-[3-(5-methyl-1,2,4-oxadiazol-3-yl)benzenesulfonyl]-2,8-diazaspiro[4.5]decane
7-fluoro-2-methyl-4-[4-(4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]quinoline
N-{1-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
4-{1-[(2,3-dimethoxyphenyl)methyl]piperidin-3-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
methyl 5-(1-benzyl-5-methyl-1H-1,2,3-triazole-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
3-(5-fluoro-2-methoxybenzoyl)-1-methylpiperidine
N-[2-oxo-4-(4-oxo-4H-chromen-3-yl)-1,2,3,4-tetrahydroquinolin-7-yl]methanesulfonamide
2-(2,4-dichlorophenoxy)-1-[3-(pyridin-3-yl)azetidin-1-yl]ethan-1-one
1,3-dimethyl-N-[2-(4-phenylpyrimidin-2-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-fluoro-4-[4-(1H-pyrazol-1-yl)phenyl]benzene-1-sulfonamide
N-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-6-methyl-2-(pyridin-3-yl)pyrimidin-4-amine
(2S)-2-amino-3-(4-hydroxyphenyl)-1-[4-(2-methoxyphenoxy)piperidin-1-yl]propan-1-one
N-(furan-2-ylmethyl)-N-(3-methylbutan-2-yl)-2-(pyridin-4-yl)pyrimidine-5-carboxamide
methyl 5-[(2,1,3-benzothiadiazol-5-ylmethyl)amino]-3-(furan-3-amido)-1-(2-methylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-(hydroxymethyl)-1-(3-propyl-1H-pyrazole-4-carbonyl)piperidin-3-ol
N-({3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
N,N-diethyl-1-[1-(3-phenylpropyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]-2,3-dihydro-1H-indene-5-carboxamide
2-(2-aminopyrimidin-5-yl)-8-methyl-N-[1-(pyridin-4-yl)propyl]quinoline-4-carboxamide
3,3-diphenyl-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]piperidine
(2R,4S)-4-hydroxy-1-[3-(methylsulfanyl)propyl]piperidine-2-carboxylic acid
1-(cyclohexylmethyl)-5-[4-(2,3-dimethylphenyl)piperazine-1-carbonyl]-N-ethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
(2R,3R,6R)-5-(2,1,3-benzoxadiazol-4-ylmethyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-oxo-S-(thiophen-2-yl)ethane-1-sulfonamido
1-(4-methylpiperazin-1-yl)-3-[1-(1-phenylpiperidin-4-yl)piperidin-3-yl]propan-1-one
N-(1-methoxypropan-2-yl)-5-methyl-6-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}thieno[2,3-d]pyrimidin-4-amine
methyl 4-[(2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}phenyl)formamido]butanoate
2-{4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-(2-methyl-1H-1,3-benzodiazol-6-yl)-3-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)urea
1-{2-[4-(4-hydroxypiperidin-1-yl)piperidine-1-carbonyl]phenyl}ethan-1-one
{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}(ethyl)[2-(1H-pyrazol-1-yl)ethyl]amine
1-[2-(3-hydroxypyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]ethan-1-one