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6-{1-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]piperidin-3-yl}-2-methyl-3,4-dihydropyrimidin-4-one
3-(2-chlorophenyl)-1-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]propan-1-one
{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(2-methyl-1,3-thiazol-4-yl)methyl]amine
{1-[7-(methylsulfanyl)-3-({[(3,4,5-trimethoxyphenyl)methyl]amino}methyl)quinolin-2-yl]piperidin-3-yl}methanol
4-({1-cyclohexyl-5-[(oxolan-2-ylmethoxy)methyl]-1H-1,2,4-triazol-3-yl}methyl)-1-methylpiperidine
5-methyl-4-[methyl(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxylic acid
1-ethyl-6-oxo-N-{[1-(phenoxymethyl)cyclopropyl]methyl}piperidine-3-carboxamide
[3-(3-methylbut-2-en-1-yl)-1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]methanol
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}pyrimidin-2-amine
N-[(3-chlorophenyl)methyl]-3-(4-methylpiperazine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(3,4-difluorophenyl)-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]acetamide
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl})amine
2-(4-{[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]methyl}phenoxy)pyrimidine
3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(1-phenylcyclopentyl)methyl]propanamide
[2-(1H-1,3-benzodiazol-2-yl)ethyl]({[6-(pyrrolidin-1-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl})amine
N-(3-chloro-4-propoxyphenyl)-4-(pyridin-4-yl)piperazine-1-carboxamide
3-[(4aR,7aS)-6,6-dioxo-4-{[4-(propan-2-yl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
1-cyclobutanecarbonyl-N-(cyclohex-1-en-1-ylmethyl)piperidine-4-carboxamide
N-[(5-{[3-(cyclopentyloxy)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
2-{4-[(2-methoxypyridin-3-yl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
N-(furan-2-ylmethyl)-1-[2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetyl]piperidine-4-carboxamide
8-benzoyl-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1R,5S)-6-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-6-azabicyclo[3.2.1]octane
(4aS,8aR)-1-[2-(pyridin-2-yl)ethyl]-6-(thiophen-2-ylmethyl)-decahydro-1,6-naphthyridin-2-one
2-{5-[(1S)-1-hydroxy-2-phenylethyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}acetic acid
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(3-methoxypropanoyl)pyrrolidin-3-yl]-2-methyl-1,3-thiazole-4-carboxamide
4-[2-(dimethylamino)-2-(3-methylphenyl)acetyl]-1-phenylpiperazin-2-one
2-cyclohexyl-5-{[4-(oxan-4-yl)piperazin-1-yl]methyl}pyrimidine
3-{2-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
(4aS,7aR)-1-[(4-fluorophenyl)methyl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(4-methoxy-2,6-dimethylphenyl)thieno[2,3-d]pyrimidine
methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]{[3-({1-[2-(trifluoromethyl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}amine
N,N-dimethyl-5-({methyl[1-(4-methyl-1,3-thiazol-2-yl)ethyl]amino}methyl)pyrimidin-2-amine
{3-propyl-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]piperidin-3-yl}methanol
2-(4,5-dimethylfuran-2-yl)-1-(prop-2-en-1-yl)-1H-imidazole
[(3S,5R)-5-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(pyridine-2-carbonyl)piperidin-3-yl]methanol
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2,5-dimethylbenzene-1-sulfonamide
1-ethyl-N-(furan-3-ylmethyl)-N-methyl-5-(morpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[4-(hydroxymethyl)phenyl]-2-[(2-methoxyethyl)(methyl)amino]acetic acid
2-(4,6-dimethylpyrimidin-2-yl)benzonitrile
1-(1H-pyrazole-4-carbonyl)-4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazine
(3R,4S)-4-(5-methylfuran-2-yl)-1-[6-(morpholine-4-carbonyl)pyrazin-2-yl]pyrrolidin-3-amine
1-(4-aminopyrimidin-2-yl)-4-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-1,4-diazepan-6-ol
3-[1-(4-methoxyphenyl)-1H-1,2,4-triazol-5-yl]pyridin-2-ol
N-(prop-2-en-1-yl)-3-[4-(trifluoromethyl)benzoyl]piperidine-1-carboxamide
(2S)-2-(methylamino)-1-{4-[4-(propan-2-yl)-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}propan-1-one
8-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
6-fluoro-4-hydroxy-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methylquinoline-3-carboxamide
2-({3-[4-(2-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol