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3-(2H-1,3-benzodioxol-5-ylmethyl)-6-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
3-cyclopropyl-5-(naphthalen-1-yl)-1H-1,2,4-triazole
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-methyl-N-[2-(oxan-4-yl)ethyl]benzamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-4-methyl-N-(oxolan-2-ylmethyl)pyrimidine-5-carboxamide
2-ethyl-4-{[4-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}pyrimidine
7-[2-(1H-imidazol-2-yl)benzoyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{1-[1-(oxolan-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenylpropanamide
2-{9-ethyl-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}-4,6-dimethylpyridine-3-carbonitrile
5-[5-(pyrrolidin-1-ylmethyl)pyridin-2-yl]pyridin-3-amine
2-amino-N-[2-(1H-imidazol-1-yl)ethyl]-N-methyl-1,3-benzothiazole-5-carboxamide
8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{2-[3-(3-chlorophenoxy)azetidin-1-yl]-2-oxoethyl}-2-azaspiro[4.4]nonan-3-one
N-[2-(pyrrolidin-1-yl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
2-[4-(3,5-dimethylphenyl)-3-oxopiperazin-1-yl]-1,3-thiazole-4-carboxamide
5-(2-chlorophenyl)-3-(1-hydroxypropan-2-yl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
8-[(5-ethylfuran-2-yl)methyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
1-(oxane-2-carbonyl)-N-(2-phenylethyl)piperidine-4-carboxamide
3-ethyl-8-{[3-(3-fluorophenyl)oxolan-3-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl 2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}acetate
ethyl 1-[(5-acetylthiophen-3-yl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylate
N-cyclopentyl-N-[(2,5-dimethoxyphenyl)methyl]-3-ethyl-4-methyl-1H-pyrazole-5-carboxamide
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyrazin-2-ylmethyl)acetamide
2-(2-fluorophenyl)-1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
3-(2-hydroxyethyl)-4-{1-[(4-methylphenyl)amino]cyclopentanecarbonyl}piperazin-2-one
(1S,5R)-3-(2-ethoxyacetyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
2-methyl-5-phenyl-N-[1-(pyrimidin-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
3,3-dimethyl-1-[(3S,4R)-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]urea
methyl 4-{4-[3-(dimethylamino)pyrazin-2-yl]piperazin-1-yl}benzoate
N-(2,4-dimethoxyphenyl)-N'-[2-(2,5-dimethylphenyl)ethyl]propanediamide
2-[5-(7-chloroquinolin-4-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
dimethyl({2-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]phenyl}methyl)amine
10-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-9-methoxy-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
2-(2H-1,2,3-benzotriazol-2-yl)-1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}ethan-1-one
5-[4-methoxy-2-(1H-pyrazol-1-yl)phenyl]pyridine-3-carboxamide
methyl 4-({[(3R,5S)-1-(propan-2-yl)-5-[(propan-2-yl)carbamoyl]pyrrolidin-3-yl]amino}methyl)benzoate
2-{[4-(2-amino-6-ethyl-5-methylpyrimidin-4-yl)piperazin-1-yl]methyl}benzonitrile
2-ethyl-N-[(1R)-2,2,2-trifluoro-1-phenylethyl]pyrimidine-5-carboxamide
2-[(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)amino]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-2-methylpropyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
3-{4-[2-(furan-2-yl)pyrrolidine-1-carbonyl]phenyl}-1H-pyrazole
N-[1-(1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]pyridine-3-carboxamide
2-[3-(naphthalene-1-carbonyl)piperidin-1-yl]propane-1,3-diol
1-(4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)piperidine-4-carboxamide
1-(4-methoxyphenyl)-3-methyl-4-(2-propoxybenzoyl)piperazin-2-one
N-(1-hydroxybutan-2-yl)-3-(1H-pyrazol-1-yl)-N-(pyridin-3-ylmethyl)benzamide
2-[2-(dimethylamino)ethyl]-8-[2-(methylamino)pyridine-4-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[4-(2-aminopyrimidin-4-yl)-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
9-(2,6-dimethylpyridin-4-yl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2,3-dichloro-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}benzamide