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3-[methyl(2-{4-[(2-methylphenyl)methyl]piperazin-1-yl}pyrimidin-4-yl)amino]propane-1,2-diol
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-{[4-(dimethylsulfamoyl)phenyl]methyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-(piperidin-3-yl)-N-[(1-propyl-1H-imidazol-2-yl)methyl]benzamide
[5-({3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)furan-2-yl]methanol
2-(morpholin-4-yl)-N4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyrimidine-4,6-diamine
8-(4-cyclobutyl-6-methylpyrimidin-2-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[2-(2-ethoxyphenyl)ethyl]-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
2,7,8-trimethyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]quinoline-4-carboxamide
(4aS,7aR)-1-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-amino-2-methyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)propanamide
({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]methylamine
1-[2,2-bis(prop-2-en-1-yl)piperidin-1-yl]-2-(2,2,3,3-tetrafluoropropoxy)ethan-1-one
2-amino-5-methyl-4-[2-(morpholin-4-yl)pyrimidin-5-yl]-6-(propan-2-yl)pyridine-3-carbonitrile
N,2,5,6-tetramethyl-N-{[1-(propan-2-yl)piperidin-3-yl]methyl}pyrimidin-4-amine
3-(2-phenylethyl)-5-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl]-1H-1,2,4-triazole
({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)(2-methoxyethyl)[(4-methylphenyl)methyl]amine
5-(azepane-1-carbonyl)-1-(butan-2-yl)-4-oxo-N-[(4-phenyloxan-4-yl)methyl]-1,4-dihydropyridine-3-carboxamide
5-{3-cyclohexyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2-ethyl-4-methyl-1,3-oxazole
N-[(4-hydroxyazepan-4-yl)methyl]-2-propyl-1,3-thiazole-4-carboxamide
N-[(3R,4R)-4-hydroxypyrrolidin-3-yl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
5-(azocane-1-carbonyl)-N-ethyl-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
3-(3-cyclohexylpropanoyl)-9-methoxy-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-[methyl(5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)amino]ethan-1-ol
6-(difluoromethyl)-2-[2-({[(5-ethylpyridin-2-yl)methyl](methyl)amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
3-(5-methyl-4H-1,2,4-triazol-3-yl)-1-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]propan-1-one
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
2-(methylsulfanyl)-5-{[4-(pyridin-4-yl)piperazin-1-yl]methyl}pyrimidine
3-(2-ethyl-1H-imidazol-1-yl)-1-[3-(3-methylphenoxy)azetidin-1-yl]propan-1-one
1-[2-hydroxy-3-(4-methoxy-2-{[methyl(2-methylpropyl)amino]methyl}phenoxy)propyl]piperidin-4-ol
11-[2-(1H-imidazol-2-yl)benzoyl]-3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane
(3S,4S)-1-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
ethyl 3-benzyl-1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidine-3-carboxylate
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[1-(4-methanesulfonylphenyl)propyl]propanamide
1-{[1-(3,3-dimethylbutanoyl)piperidin-3-yl]methyl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
methyl 2-(8-{[5-(methoxymethyl)furan-2-yl]methyl}-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl)acetate
2-(1-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)-1,3-benzoxazole
1-({5-[(2,3-difluoro-4-methylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-[4-(4-methylphenyl)-1H-pyrazol-1-yl]acetamide
N3-ethyl-1-(2-methylpropyl)-4-oxo-N5-(3-phenylpropyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-3-(4H-1,2,4-triazol-4-yl)propanamide
4-[(4-fluorophenyl)methyl]-3-(2-oxo-2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethyl)piperazin-2-one
N-[(3R,4S)-1-acetyl-4-propylpyrrolidin-3-yl]-4-methoxypiperidine-1-sulfonamide
5-(1-{4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]-1H-1,2,3-triazol-1-yl}ethyl)-1H-1,2,3,4-tetrazole
2-({4-[4-methoxy-3-(trifluoromethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethan-1-ol
8-benzyl-3-(2-methylpropyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(2,4-dichloro-6-methylphenyl)methyl]-5-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(1S,5R)-3-[(2-fluoro-4-methoxyphenyl)methyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-(3-fluorophenoxymethyl)-N-[(2-methoxyphenyl)methyl]-N-methyl-1H-pyrazole-3-carboxamide