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(2S,4R)-1-[(3-chlorophenyl)methyl]-N-(propan-2-yl)-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
8-(2-amino-6-methoxypyrimidin-4-yl)-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}-2-[3-(methylsulfanyl)phenyl]acetic acid
1-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-3-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}urea
4-{5-[1-(furan-2-ylmethyl)piperidin-3-yl]-1,2,4-oxadiazol-3-yl}pyridine
N-methyl-N-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)thian-4-amine
1-cyclopentanecarbonyl-3-[2-(3-fluorophenyl)ethyl]piperidine
1-[(3-hydroxyphenyl)methyl]-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
(3S,4S)-1-[(3-chloro-4-methoxyphenyl)methyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
2-amino-7-(quinoxaline-5-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-4-(3-hydroxy-3-methylbutyl)benzamide
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-{[(2,5-difluorophenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
5-methyl-N,N-bis(1,3-oxazol-4-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
2-ethyl-1-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}butan-1-one
2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-3-carbonitrile
6-fluoro-2-({[3-(4-methylpiperazin-1-yl)propyl]amino}methyl)quinolin-4-ol
6-chloro-3-fluoro-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}imidazo[1,2-a]pyridine-2-carboxamide
N-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-3-(1H-1,2,4-triazol-1-yl)adamantan-1-amine
N,1-dimethyl-N-{1-[1-(2-methylpyridine-3-carbonyl)piperidin-4-yl]-2-phenylethyl}-1H-pyrazole-3-carboxamide
2-ethyl-4-phenyl-9-(2-propoxyacetyl)-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-4-(2-methylphenyl)-1-(3-propyl-1H-pyrazole-5-carbonyl)piperazine
1-{[2-(ethylamino)pyrimidin-5-yl]methyl}-4-(1H-imidazole-2-carbonyl)-1,4-diazepan-6-ol
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
1-{3-fluoro-8-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-(4-methoxyphenyl)-2-methylpiperazine
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-4-(pyridin-3-yl)pyrimidin-2-amine
N-[3-(4-fluorophenyl)phenyl]-1-(thian-4-yl)piperidine-3-carboxamide
5-(1H-indole-3-carbonyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
methyl 4-[2-(2,3-difluoro-4-methoxyphenyl)-1H-imidazol-1-yl]butanoate
N4,N4-dimethyl-6-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrimidine-2,4-diamine
1-(2,3-difluoro-4-methoxybenzoyl)-3-(2-ethylphenoxy)azetidine
N-(butan-2-yl)-3-(methylsulfanyl)-N-(pyridin-4-ylmethyl)propanamide
{5-fluoro-7-[2-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
5-ethyl-N4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N4-methylpyrimidine-2,4-diamine
2-(4-{[4-(dimethylcarbamoyl)piperazin-1-yl]methyl}-2-methoxyphenoxy)propanoic acid
4-({2-[1-(pyrrolidine-1-sulfonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
4-[(4-chlorophenyl)methyl]-1-(9H-purin-6-yl)piperidine-4-carboxylic acid
N-(2-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)acetamide
methyl 2-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}butanoate
2-(1H-indole-5-carbonyl)-6-methyl-5-(5-methyl-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine
7-(cyclobutylmethyl)-2-(1-methyl-1H-pyrazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-[2-({2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}amino)pyrimidin-4-yl]piperidin-3-ol
2-(2-ethyl-1H-imidazol-1-yl)-1-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]ethan-1-one
[(dimethyl-1,3-thiazol-5-yl)methyl](ethyl)[2-(morpholin-4-yl)ethyl]amine
(3R,4R)-1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]oxane-4-carboxamide
N-[2-(thiophen-2-yl)ethyl]-2-(trifluoromethyl)pyrimidin-4-amine
methyl (2S,4S)-4-(3-chloro-4-fluoro-1-benzothiophene-2-amido)-1-methylpyrrolidine-2-carboxylate
(1S,5R)-6-(1,3-thiazol-4-ylmethyl)-3-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(2S,4R)-1-[(2-aminopyridin-3-yl)methyl]-4-(3-hydroxybenzamido)-N-methylpyrrolidine-2-carboxamide
(5S,9aS,9bS)-5-[2-(furan-2-yl)phenyl]-2-(1-methylpiperidin-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one