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methyl 2-[(2,3-dimethylphenyl)sulfamoyl]-6-(2,2-dimethylpropanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(methoxymethyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]cyclobutane-1-carboxamide
5-{[4-(3-methoxybenzoyl)piperazin-1-yl]methyl}-2-(methylsulfanyl)pyrimidine
1-[(2,4-dimethyl-5-{1-propyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)methyl]-1H-1,2,4-triazole
3-({1-[5-(1-ethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]propan-2-yl}oxy)pyridine
4-(4-chlorophenyl)-N-[1-(methoxymethyl)cyclopentyl]butanamide
1-{[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
8-fluoro-N-{2-hydroxy-2-[2-(trifluoromethyl)phenyl]ethyl}quinoline-2-carboxamide
1-cyclohexyl-N-cyclopropyl-5-{4-[(3-methoxyphenyl)methyl]piperazine-1-carbonyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
3-[hydroxy(phenyl)methyl]-4-(pyridin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,4S)-4-[2-(carbamoylamino)acetamido]-1-[(3-ethenylphenyl)methyl]-N-ethylpyrrolidine-2-carboxamide
N-benzyl-2-cyclopentyl-N-(1,3-thiazol-2-ylmethyl)acetamide
4-[1-(1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-4-yl)ethyl]morpholine
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(pyridin-4-ylmethyl)-1,4-diazepane
{4-[(4-{5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}-1H-1,2,3-triazol-1-yl)methyl]phenyl}methanol
ethyl 2-(5-{1-[({2-[(3-fluorophenyl)methoxy]-6-methylquinolin-3-yl}methyl)amino]ethyl}-4H-1,2,4-triazol-3-yl)acetate
3-{[(4aS,7aR)-4-[(4-methyl-1H-imidazol-5-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}benzonitrile
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2,5,6-trimethyl-N-[3-(pyridin-3-yloxy)propyl]pyrimidin-4-amine
2-(morpholin-4-yl)-2-(pyridin-3-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)acetamide
1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-4-(4-methylphenoxy)piperidine
N-methyl-2-[4-(propan-2-yl)morpholin-2-yl]-N-(thiophen-3-ylmethyl)acetamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[(3-fluorophenyl)methyl]-1-(2-methylpropyl)piperidine-3,5-dicarboxamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(2-methylpropanoyl)piperidine-2-carboxamide
4-[5-(3-benzoylpiperidine-1-carbonyl)-1H-pyrazol-3-yl]pyridine
N-propyl-5-{[4-(pyridin-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyrimidin-2-amine
2-(prop-2-en-1-yl)-9-(pyrazine-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(3,3-diphenylpiperidin-1-yl)-2-(1H-imidazol-1-yl)propan-1-one
1-[2-methoxy-4-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
2-{2-[2-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]ethyl}-1H-1,3-benzodiazole
N-[(5-methylfuran-2-yl)methyl]-3-[1-(oxan-4-yl)piperidin-3-yl]propanamide
N-({6-[4-(pentan-3-yl)piperazin-1-yl]pyridin-3-yl}methyl)acetamide
4-[4-(4-hydroxy-3-methoxybenzoyl)-2-oxopiperazin-1-yl]benzonitrile
2-methyl-4-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazole
N-(2-methylpropyl)-1-[(1s,4s)-4-[3-(pyridin-3-yl)propanamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-[6-(morpholin-4-yl)pyrimidin-4-yl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-acetamido-3-hydroxypropanamide
6-[2-(3,4-dichlorophenyl)morpholin-4-yl]-N-ethyl-N-methylpyridine-3-carboxamide
{1-[({[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)methyl]cyclobutyl}methanol
N,4-dimethyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,2,5-oxadiazole-3-carboxamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
4-hydroxy-2-(pyridin-2-yl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]pyrimidine-5-carboxamide
1-[5-(azepan-1-ylmethyl)-2-methoxyphenoxy]-3-(piperidin-1-yl)propan-2-ol
1-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-4-(1,3-thiazol-2-yl)piperazine
1-{2-hydroxy-3-[2-methoxy-4-({[(5-methylthiophen-2-yl)methyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
3-cyclopentaneamido-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)benzamide
ethyl 3-[(2,4-difluorophenyl)methyl]piperidine-3-carboxylate
6-[(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(4,6-dimethyl-1-benzofuran-3-yl)-N-[2-(2-methylpropanesulfonyl)ethyl]acetamide
N-[(1S,2R)-2-aminocyclobutyl]-1-[(4-methoxyphenyl)amino]cyclopentane-1-carboxamide