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2-(pyridin-4-ylmethyl)-9-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N4-(thiolan-3-yl)-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
2,2-dimethyl-N-(1-{1-[3-(2-methyl-1H-1,3-benzodiazol-1-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
(3S,9aR)-3-[(2S)-butan-2-yl]-8-(2,4,5-trifluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-cyclohexyl-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxamide
N-[(5-methylfuran-2-yl)methyl]-3-[(oxolan-3-yl)sulfamoyl]benzamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-(pentan-3-yl)acetamide
6-[({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(2,3-dimethoxyphenyl)methyl]amino}-N-[2-(2-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
2-(4-{1-[(3-methyl-1H-pyrazol-5-yl)methyl]-4-phenyl-1H-imidazol-5-yl}phenoxy)ethan-1-ol
2-(2,5-dimethylphenoxy)-N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]propanamide
2-[5-methoxy-2-(prop-2-yn-1-yloxy)phenyl]-6-methyl-1H-1,3-benzodiazole
6-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-4-methyl-1,3-benzothiazol-2-amine
(2S,4R)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-4-(thiophene-2-amido)pyrrolidine-2-carboxamide
5-[4-(4-fluorophenoxy)piperidine-1-carbonyl]-1H-indole
4-{[2-(3,4-dichlorophenyl)morpholin-4-yl]methyl}-2,6-dimethoxyphenol
3-(3,4-difluorophenyl)-5-[(5-propylfuran-2-yl)methyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-[3-(3-benzyl-1H-1,2,4-triazol-5-yl)phenyl]-5-methyl-1H-1,2,3,4-tetrazole
2-{[(3R,5S)-5-[4-(adamantan-2-yl)piperazine-1-carbonyl]-1-benzylpyrrolidin-3-yl]sulfanyl}pyrimidine
2-{[3-(naphthalene-1-carbonyl)piperidin-1-yl]methyl}phenol
1-methyl-6-oxo-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}-1,6-dihydropyridazine-3-carboxamide
4-ethyl-1-[2-(phenylsulfanyl)ethyl]-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{[4-({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}(methyl)amino)-6-methylpyrimidin-2-yl]amino}phenol
(2R,3R)-3-amino-1'-(1-methyl-1H-indole-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(pyrimidin-2-yl)-1,4-diazepane
(1S,5R)-3-(2-methylpropanoyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-3-ethyl-N,5-dimethyl-1,2-oxazole-4-carboxamide
7-fluoro-3-{[(2-hydroxy-2-phenylethyl)(methyl)amino]methyl}-1-[(3-methoxyphenyl)methyl]-1,2-dihydroquinolin-2-one
1,6-dimethyl-N-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H-indole-2-carboxamide
N-ethyl-1-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
1-(2H-1,3-benzodioxol-4-ylmethyl)-3-[3-(trifluoromethyl)benzoyl]piperidine
6-fluoro-2-({[1-(pyridin-4-yl)propyl]amino}methyl)quinolin-4-ol
2-amino-N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)acetamide
N-(furan-2-ylmethyl)-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
(1-{[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]methyl}cyclobutyl)methanol
N-[(1-propyl-1H-imidazol-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-cyclopentyl-4-[4-({2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}amino)piperidin-1-yl]benzamide
4-(azetidin-1-ylmethyl)-1-[4-(propan-2-yl)phenyl]-1H-pyrazole
6-{4-[1-(methoxymethyl)cyclobutanecarbonyl]piperazin-1-yl}pyridine-3-carbonitrile
(3S,7S,8aS)-7-({[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)-3-propyl-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-{2-[3-(2-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}-3-methylimidazolidin-2-one
3-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-1-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-4-yl}urea
({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)(oxolan-2-ylmethyl)(thiophen-3-ylmethyl)amine
1-(3-{[3-(1,2-oxazinane-2-carbonyl)-1H-pyrazol-5-yl]methoxy}phenyl)ethan-1-one
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-ethyl-1,2-oxazole-5-carboxamide
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-3-ethoxypropan-1-one
2-(3-chloropyridin-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
5-hydroxy-N-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}pyrazine-2-carboxamide
3-hydroxy-3-[({imidazo[1,2-a]pyridin-2-ylmethyl}amino)methyl]-1-(2-phenylethyl)piperidin-2-one
2-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-N,N-dimethylacetamide