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3-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-1-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}urea
1-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(methoxymethyl)piperidine
2-(oxolan-2-ylmethoxy)-1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]ethan-1-one
1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-4-(pyridin-4-yl)-1,4-diazepane
(3R)-1-({1-[(1-cyclohexanecarbonylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}methyl)pyrrolidin-3-amine
1-(cyclopropanesulfonyl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-(3-chloro-4-methoxyphenyl)-6-[2-(pyridin-4-ylsulfanyl)acetyl]-6-azaspiro[2.5]octane-1-carboxamide
N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-3-(piperidin-3-yl)benzamide
6-{[1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
N-cyclobutyl-3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
3-{1-methyl-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl}-1H-indazole
4-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1-(2-methoxyethyl)pyrrolidin-2-one
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-6-methylpyridine-3-carboxamide
1-{2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-(furan-2-ylmethyl)-N-methylpiperidine-3-carboxamide
5-methoxy-1-methyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1H-indole-2-carboxamide
3-(4-benzyl-3-ethyl-5-oxo-1,4-diazepane-1-carbonyl)-5-fluorobenzonitrile
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
N-cyclohexyl-N-methyl-2-(5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)acetamide
N-[(3S,4R)-1-[2-(5-ethyl-1-benzofuran-3-yl)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
(3aS,6aS)-2-cyclobutanecarbonyl-5-[2-(2,3-dimethylphenoxy)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,4-dichlorophenyl)urea
2-[1-(1-phenyl-1H-1,2,3-triazole-5-carbonyl)pyrrolidin-2-yl]pyridine
5-ethyl-2-methyl-4-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
N-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]pyrazolo[1,5-a]pyridine-7-carboxamide
N-[1-(1-benzyl-3-phenyl-1H-1,2,4-triazol-5-yl)ethyl]methanesulfonamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]acetamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-(1H-indazol-3-ylformamido)acetic acid
1-[(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methylpyrrolidine-3-carbonyl]-1,4-diazepan-5-one
4-[2-(2-aminoethyl)morpholin-4-yl]-N-cyclopropyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
4-cyclopropyl-6-[3-(1-methoxyethyl)phenyl]pyrimidine
N-(1-hydroxy-2-methylpropan-2-yl)-5-methyl-4-{[3-(morpholin-4-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
3-(3-chloro-1,2-oxazol-5-yl)-1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}propan-1-one
N-(1-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
(3aR,5S,6S,7aS)-2-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-octahydro-1H-isoindole-5,6-diol
1-(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazin-1-yl)-2-phenoxyethan-1-one
(1-benzofuran-2-ylmethyl)(ethyl)(oxan-4-ylmethyl)amine
1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-2-[methyl(pyridin-2-ylmethyl)amino]ethan-1-one
1-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-4-phenoxypiperidine-4-carboxylic acid
1-{3-carboxy-5-[(propan-2-yl)sulfamoyl]phenyl}-1H-pyrazole-4-carboxylic acid
3-(5-benzyl-1,3,4-thiadiazol-2-yl)-1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)urea
3-{7-methylthieno[3,2-d]pyrimidin-4-yl}-1H-pyrazole
(4-{[(3-ethoxy-4-methoxyphenyl)methyl](methyl)amino}quinazolin-2-yl)methanol
1-{[(3R,4R)-4-(hydroxymethyl)-1-(5-methoxyfuran-2-carbonyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-methyl-1,2,3-thiadiazole-5-carboxamide
(1S,5R)-3-methyl-6-(7-methyl-1-benzofuran-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
6,8-dimethyl-3-({methyl[(3-methylpyridin-2-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
1-{5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}azepane
3-hexyl-8-(4-methylpyrimidine-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]benzene-1,3-diol