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(4aS,8aR)-6-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
6-ethyl-N-(1-methanesulfonylpiperidin-4-yl)-4-methylquinolin-2-amine
4-(4-{1-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
N,N-bis(prop-2-en-1-yl)-2-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]acetamide
8-[(1R,2R,3S,4S)-3-aminobicyclo[2.2.1]heptane-2-carbonyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-(2,6-difluorophenoxymethyl)-N-[(3-fluoro-4-methylphenyl)methyl]-1,2-oxazole-3-carboxamide
N-[(4-methoxyphenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
8-(5-phenyl-1,2,4-oxadiazol-3-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-fluorobenzamide
3-{1-[3-(pyridin-3-yloxy)propyl]-1H-imidazol-2-yl}phenol
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]pyrrolidine-1-sulfonamide
1-[(3,4-difluorophenyl)methyl]-3-({[2-(furan-2-yl)ethyl]amino}methyl)-3-hydroxypiperidin-2-one
methyl 2-{8-[(3-hydroxyphenyl)methyl]-1-(2-methoxyethyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
4-[1-(2-methoxyphenyl)-3-(propan-2-yl)-1H-1,2,4-triazole-5-carbonyl]morpholine
N-(but-2-yn-1-yl)-1-[(2-fluorophenyl)methyl]-N-(furan-2-ylmethyl)-6-oxopiperidine-3-carboxamide
5-[1-(furan-2-ylmethyl)pyrrolidin-2-yl]-N-(1,3-thiazol-2-yl)thiophene-2-carboxamide
6-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]pyridine-2-carbonitrile
3-(1-{2-[4-(methylsulfanyl)phenyl]acetyl}piperidin-3-yl)-1-(morpholin-4-yl)propan-1-one
N-{[(3S,4S)-3-hydroxy-1-[(2-methoxy-4-methylphenyl)methyl]piperidin-4-yl]methyl}cyclopropanecarboxamide
4-[3-(furan-2-yl)-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]-1-(2-methoxyethyl)pyrrolidin-2-one
N-[2-(methylsulfanyl)phenyl]-N'-(pyridin-2-ylmethyl)butanediamide
4-{4-[2-(2,5-dimethoxyphenyl)acetyl]piperazin-1-yl}-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-[2-(1-benzylpyrrolidin-3-yl)ethyl]-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-methyl-4-{1-[1-(3-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]ethyl}piperazine
1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
5-[3-(methoxymethyl)piperidine-1-carbonyl]-N-(propan-2-yl)pyridin-2-amine
N-{1-[3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]ethyl}-6-(methoxymethyl)pyrimidin-4-amine
5-(5-methylfuran-2-yl)-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-1,2,4-triazin-3-amine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-(pyridin-2-ylmethyl)piperidin-3-amine
2-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]pyrimidin-4-amine
1-(methoxymethyl)-N-{1-[(3-methylphenyl)methyl]cyclopropyl}cyclobutane-1-carboxamide
2-{[(4aR,8aR)-4a-hydroxy-7-methanesulfonyl-decahydro-2,7-naphthyridin-2-yl]methyl}-5-methoxy-4H-pyran-4-one
3-{2-[2-(3-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-5,5-dimethyl-1,3-oxazolidine-2,4-dione
6-[3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]pyridine-2-carbonitrile
4-hydroxy-N-[2-(4-methoxyphenyl)ethyl]-2-methyl-N-(oxolan-2-ylmethyl)pyrimidine-5-carboxamide
3-({1-[3-(1,3-thiazol-4-yl)phenyl]piperidin-4-yl}amino)-2,3-dihydro-1λ6-thiophene-1,1-dione
6-(2H-1,3-benzodioxole-5-carbonyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
(3S,4S)-4-cyclopropyl-1-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}pyrrolidine-3-carboxylic acid
3-({4-phenyl-5-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H-imidazol-1-yl}methyl)-5-(propan-2-yl)-1,2,4-oxadiazole
N-butyl-7-[(3,4-difluorophenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)-1-azabicyclo[2.2.2]octane
3-methyl-5-(4-{[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)pyridine
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)-N-methylacetamide
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1-(oxan-4-yl)piperidine-3-carboxamide
N-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-1-(4-fluorophenyl)piperidin-4-amine
(2R,3R,6R)-N-tert-butyl-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]-1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethan-1-one
1-{3-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(5-{[5-(oxan-2-yl)thiophen-2-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl)pyridine
N-(furan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-2,3-dihydro-1H-indene-1-carboxamide