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N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-3-(1H-pyrazol-4-yl)benzamide
(3S)-3-ethyl-4-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}morpholine
4-({[1-(1-methylpiperidin-4-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)pyridine
N-[(2R,3R)-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(pyridin-3-yl)acetamide
4-[3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine-1-carbonyl]-1,2-dihydrophthalazin-1-one
4-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-3-(pyrrolidin-3-yl)benzamide
N-[(1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidin-3-yl)methyl]-1,2,5-oxadiazole-3-carboxamide
methyl 2-[butyl(methyl)sulfamoyl]-6-[(5-chloro-2-hydroxyphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-ethyl-1'-[6-(trifluoromethyl)pyridin-2-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{9-[(2-fluorophenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
[1-(2-{4-phenyl-5-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-1-yl}ethyl)piperidin-2-yl]methanol
2-{[3-({[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}carbamoyl)phenyl]amino}acetic acid
4-{[2-methyl-5-(trifluoromethyl)phenyl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1-(furan-2-ylmethyl)-N-methylpiperidine-3-carboxamide
N-(3,5-dimethylphenyl)-N'-(prop-2-en-1-yl)-N'-(pyridin-3-ylmethyl)propanediamide
2,7-dioxo-N-{2-[3-(trifluoromethyl)phenyl]ethyl}-1,3-diazepane-4-carboxamide
(2R)-2-amino-1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-(ethylsulfanyl)propan-1-one
4-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-4H-1,2,4-triazole
N,6-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4-oxo-4H-pyran-2-carboxamide
N-{2-[2-(1H-imidazol-4-yl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}-1-phenylcyclopropane-1-carboxamide
1-(but-2-yn-1-yl)-3-[3-(4-methanesulfonylphenyl)phenyl]-1H-pyrazole
1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
3-{1-[1-(thiophene-2-sulfonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-1-ol
N-[3-(3-carbamoylpiperidin-1-yl)propyl]-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyrazine-2-carboxamide
N-cyclopentyl-1-methyl-5-(thiolan-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(4-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methoxy}phenyl)-1H-1,3-benzodiazole
(3S,4R)-1-(5-{[(4,6-dimethylpyrimidin-2-yl)sulfanyl]methyl}furan-2-carbonyl)-4-methylpiperidine-3,4-diol
4-(2-benzyl-3-oxopiperazine-1-carbonyl)pyridin-1-ium-1-olate
1-{2,7-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4-(pyridin-2-yl)piperidin-4-ol
4-(6-aminopyridine-3-carbonyl)-5-butyl-1-(3-methylphenyl)piperazin-2-one
3-[1-(6-methoxy-3-methyl-1-benzofuran-2-yl)-N-(pyridin-3-ylmethyl)formamido]propanoic acid
methyl 3-chloro-4-({9-oxa-2-azaspiro[5.5]undecane-2-carbonyl}amino)benzoate
4-[(2S)-1-[4-(5-methylfuran-2-yl)benzoyl]pyrrolidine-2-carbonyl]morpholine
2-[4-({2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}amino)pyrimidin-5-yl]acetic acid
1-{1-[(3,5-dimethoxyphenyl)methyl]piperidin-4-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
1-(2-methoxyethyl)-1-(oxolan-2-ylmethyl)-3-(trimethyl-1H-pyrazol-4-yl)urea
2-{[6-amino-2-(benzylsulfanyl)pyrimidin-4-yl]amino}ethan-1-ol
2-(3-methoxypropyl)-8-(5-methyl-1,2-oxazole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
5-{[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]carbonyl}-1,2-dihydropyridin-2-one
N-{[7-chloro-2-(dimethylamino)quinolin-3-yl]methyl}-3,5-dimethoxy-N-(2-methoxyethyl)benzamide
1-[1-(pyridin-3-ylmethyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-(pyridin-2-ylmethyl)piperidine-4-carboxylic acid
4-ethyl-5-methyl-N-{1-oxaspiro[4.4]nonan-3-yl}pyrimidin-2-amine
2-methoxy-1-[1'-(4-methoxybenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
5-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1S,6R)-3-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-3,9-diazabicyclo[4.2.1]nonane
4-(4-{[3-(2-hydroxyethyl)-4-(3-phenylpropyl)piperazin-1-yl]methyl}phenyl)but-3-yn-1-ol
1-[(4aR,8aS)-1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-decahydro-1,6-naphthyridin-6-yl]-2-phenylethan-1-one