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N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-4-methoxybenzene-1-sulfonamide
1-[7-(1-methyl-1H-pyrazole-3-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]azepane
4-{3-[2-(furan-2-yl)-1H-imidazol-1-yl]phenyl}-2-methylpyrimidine
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-1,2,3-triazole-5-carboxamide
6-ethyl-2-methyl-4-[2-(1H-pyrazol-1-ylmethyl)pyrrolidine-1-carbonyl]quinoline
4-benzyl-3-ethyl-1-(2-hydroxyethyl)-1,4-diazepan-5-one
2-ethyl-N-(1-ethyl-4-methyl-1H-pyrazol-5-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
6-(methoxymethyl)-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]pyrimidin-4-amine
1-{2-[(dimethylamino)methyl]benzoyl}-N-(4-fluorophenyl)piperidin-3-amine
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
3-butyl-1-methyl-4-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}piperazin-2-one
methyl[3-(5-methylfuran-2-yl)butyl]{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amine
5-{[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]methyl}-2,1,3-benzoxadiazole
4-{[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]methyl}-5-(hydroxymethyl)-2-methylpyridin-3-ol
N-{[4-(2-methoxyethoxy)phenyl]methyl}-4-(piperidin-3-yl)benzamide
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methylacetamide
1-(5-cyano-2-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
2-amino-6-(propan-2-yl)-4-[2-(propylamino)pyrimidin-5-yl]pyridine-3-carbonitrile
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)but-3-enamide
2-[(4-methylquinolin-2-yl)sulfanyl]-N-[(6-oxo-1,6-dihydropyrimidin-4-yl)methyl]propanamide
1-[(1s,4s)-4-aminocyclohexyl]-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
8-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
7-(oxan-4-yl)-2-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(1H-imidazol-1-yl)butan-1-one
4-ethyl-3-[(1-{[2-(methylamino)pyridin-3-yl]methyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-6-methyl-4-oxo-2-propyl-N-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
1-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-[(3-methylphenyl)sulfanyl]piperidine
3-cyano-N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-5-fluorobenzamide
2-(2-oxo-2,3-dihydro-1H-imidazole-4-carbonyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
(2R,6S)-2,6-dimethyl-4-{2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carbonyl}morpholine
5-{1-[4-(2,3-dihydro-1H-isoindol-2-yl)butanoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]pyrimidine-5-carboxamide
[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl](methyl)[1-(pyridin-3-yl)ethyl]amine
N,2-dimethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}quinolin-4-amine
N-[(3-methyl-1-benzofuran-2-yl)methyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
N,N-dimethyl-6-[3-(1H-pyrazol-3-yl)phenyl]pyrimidin-4-amine
6-butyl-2-(2-{[4-(dimethylamino)piperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
(2S,4S)-N-ethyl-4-(2-fluorobenzamido)-1-(oxan-4-yl)pyrrolidine-2-carboxamide
8-{5-[3-(2-methyl-1H-imidazol-1-yl)propyl]-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl}quinoline
2-[4-(4-methanesulfonylphenyl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-pyrazol-5-yl)acetamide
2-methyl-8-{2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetyl}-2,8-diazaspiro[4.5]decan-3-one
(1S,2R)-N1-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-N2-propylcyclohexane-1,2-dicarboxamide
7-(ethanesulfonyl)-N2,N2,N4,N4-tetramethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperazine
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-3-(1,2-oxazinan-2-yl)propanamide
(5S)-5-[({[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}(pyridin-3-ylmethyl)amino)methyl]pyrrolidin-2-one
6-{8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecane-2-carbonyl}-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[1-(furan-2-yl)ethyl]-5-(4-methoxyphenyl)-N-methyl-1H-pyrazole-3-carboxamide
6-(thiomorpholin-4-yl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-4-one
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)benzamide