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(3S,4S)-1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-propylpyrrolidine-3-carboxylic acid
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]oxolane-3-carboxamide
2-methoxy-1-[9-(4-propylpiperazin-1-yl)-3-azaspiro[5.5]undecan-3-yl]ethan-1-one
N-[3-(cyclopentyloxy)propyl]-2-(1H-imidazol-2-yl)benzamide
2-ethyl-4-methyl-5-{1-[(4-phenyloxan-4-yl)methyl]-1H-imidazol-2-yl}-1H-imidazole
N2-phenyl-N5-propyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2,5-dicarboxamide
N-ethyl-6-[methyl(2-methylprop-2-en-1-yl)amino]-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridine-3-carboxamide
4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(5-methylthiophene-3-carbonyl)piperidine
3-(5-ethyl-1,3,4-thiadiazol-2-yl)-1-[3-(5-methyl-2H-1,2,3,4-tetrazol-2-yl)adamantan-1-yl]urea
2-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2,7-diazaspiro[4.5]decane
2-(6-methoxynaphthalen-2-yl)-4-[(1-methylpiperidin-4-yl)methyl]morpholine
2-(4-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-1-(2-phenylethyl)piperazin-2-yl)ethan-1-ol
N-cyclopentyl-1-(2-hydroxyethyl)-N-[(5-methylthiophen-2-yl)methyl]piperidine-4-carboxamide
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(4-carbamoyl-2-methylphenyl)-3-(2-methylpiperidin-1-yl)azetidine-1-carboxamide
(3E)-N-[(4-chlorophenyl)methyl]-N-ethylpent-3-enamide
5-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridin-3-amine
N4-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}pyrimidine-2,4-diamine
{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}(2-phenylethyl)amine
5-(2,6-difluorophenoxymethyl)-N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1,2-oxazole-3-carboxamide
N-(2-methoxyethyl)-5-[1-(4-methoxyphenyl)-1H-1,2,4-triazol-5-yl]-1-methyl-1H-1,3-benzodiazol-2-amine
2-{3-[(4-fluorophenyl)methoxy]phenyl}-6-(pyrrolidine-1-carbonyl)pyrazine
5-{3-[1-(1,3-thiazol-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidine
(1R,3S)-3-methoxy-7-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]-7-azaspiro[3.5]nonan-1-ol
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(pyridin-3-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
9-(3-ethyl-1,2-oxazole-5-carbonyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(1R,5R)-6-benzyl-3-(6-methylpyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(7-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]pyridine-2-carboxamide
2-[3-({4-[5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
1-methyl-3-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-5-yl)-1-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)urea
(3R,4R)-1-[(2-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-ol
3-(2-ethylphenoxy)-1-(4-methanesulfonylbenzoyl)azetidine
N-tert-butyl-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-[2-(4-chlorophenyl)-2-(piperidin-1-yl)ethyl]-5-ethyl-1,2-oxazole-3-carboxamide
N-{1-[(3-chlorophenyl)methyl]-3-methyl-1H-pyrazol-5-yl}-6-hydroxy-1,4-oxazepane-4-carboxamide
1-(4-methylphenyl)-4-{[1-(propan-2-yl)piperidin-4-yl]amino}pyrrolidin-2-one
N-{2-[1-(2,6-difluorobenzenesulfonyl)piperidin-2-yl]ethyl}acetamide
2-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrazine
4-({2-[2-(4-methanesulfonylphenyl)-1H-imidazol-1-yl]phenyl}methyl)morpholine
5-ethyl-3-{[2-(4-methoxynaphthalen-1-yl)-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole
1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
N-[4-ethoxy-3-(1H-pyrrol-1-yl)phenyl]-1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carboxamide
{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}(methyl)(2-phenoxyethyl)amine
2-(4-{[3-(morpholin-4-yl)azetidin-1-yl]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
2-amino-4-(1-methyl-1H-imidazol-5-yl)-6-[2-(trifluoromethyl)phenyl]pyridine-3-carbonitrile
N-({1-[3-(furan-2-yl)propanoyl]piperidin-3-yl}methyl)-1-phenylmethanesulfonamide
N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]pyridine-3-carboxamide
1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
2-(ethylamino)-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]pyrimidine-5-carboxamide
(4aS,8aR)-6-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one