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{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[(1-methyl-1H-pyrazol-4-yl)methyl]amine
5-[3-(2-fluorophenoxymethyl)piperidine-1-carbonyl]-2-(propan-2-yl)-1,3-benzoxazole
3-fluoro-4-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridine
1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
4-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-(oxolan-2-ylmethyl)-N-propylbutanamide
3-{1-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}phenol
N-({1-[(3-phenyl-1,2-oxazol-5-yl)methyl]pyrrolidin-3-yl}methyl)acetamide
N-methyl-3-[1-(propane-1-sulfonyl)piperidin-3-yl]-N-[2-(pyridin-2-yl)ethyl]propanamide
1-[(2-phenyl-1,3-oxazol-4-yl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
7,8-dimethyl-3-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3,4-dihydroquinazolin-4-one
2-(dimethyl-1,3-thiazol-5-yl)-N-{3-[methyl(phenyl)amino]propyl}acetamide
N-(2,3-dihydro-1H-inden-2-yl)-2-fluoro-N-methyl-5-sulfamoylbenzamide
6-methoxy-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}pyrimidin-4-amine
1,3-dimethyl-N-[(2R)-pyrrolidin-2-ylmethyl]-1H-indole-2-carboxamide
N-[3-(methylsulfanyl)propyl]-3-sulfamoylbenzamide
[3-(1H-indazol-1-yl)propyl]({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
3-benzyl-7-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-[(3R,4R)-3-hydroxy-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl]pyridine-2-carboxamide
2-(2-hydroxyethyl)-9-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)naphthalene-1-carboxamide
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
3-fluoro-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
N-(furan-2-ylmethyl)-1-methyl-N-(3-methylbutan-2-yl)-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
1-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(methylsulfanyl)ethan-1-one
N-benzyl-2,3-difluoro-N-(3-hydroxy-2-methylpropyl)-4-methylbenzamide
7-methoxy-N-(oxan-4-yl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-[1-(4-chlorophenyl)cyclobutanecarbonyl]-4-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,4-diazepan-5-one
3-[3-(4-methanesulfonylphenyl)propyl]pyridine
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]acetamide
4-(5-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
N-[2-(dimethylamino)ethyl]-1-{1-[(4-methoxy-2,5-dimethylphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
2-{[4-(2-methoxyquinolin-3-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}acetic acid
methyl 4-[7-(cyclohexylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-4-oxobutanoate
[1-({1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]methanamine
2-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}acetic acid
2-{4-[2-(4-chloro-1-methyl-1H-indazol-3-yl)-1H-imidazol-1-yl]-3,5-dimethyl-1H-pyrazol-1-yl}ethan-1-ol
2-[2-(3-methoxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]-6-methylpyridine-3-carbonitrile
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[(5-methylfuran-2-yl)methyl]pyrrolidin-3-yl]methanol
4-{5-[1-(1-ethyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]thiophene-2-carbonyl}morpholine
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-4-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]-1,3-oxazole
1-[4-(aminomethyl)phenyl]-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
2-[2-oxo-2-(3-oxo-4-phenylpiperazin-1-yl)ethyl]-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
1-{[(2R,5S)-5-(2H-1,3-benzodioxol-5-ylmethyl)oxolan-2-yl]methyl}piperidine-4-carboxylic acid
4-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}-2,1,3-benzoxadiazole
1-{5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carbonyl}-2-(3-methoxyphenyl)pyrrolidine
1-cyclopentanecarbonyl-N-[1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]piperidine-4-carboxamide
5-methyl-4-(1-methyl-1H-pyrazol-4-yl)-N-[(5-methyl-2-phenyl-2H-1,2,3-triazol-4-yl)methyl]pyrimidin-2-amine
(1R,3S)-7-(furan-3-ylmethyl)-3-methoxy-3-methyl-7-azaspiro[3.5]nonan-1-ol
1-(1-hydroxycyclopentanecarbonyl)-4-(2-methylphenoxy)piperidine-4-carboxylic acid