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N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)oxolane-3-carboxamide
2-fluoro-N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]-5-sulfamoylbenzamide
1,3-dimethyl-N-[3-(pyridin-2-yl)propyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-[2-(azepan-1-yl)ethyl]-N,1-diethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-(2-methyl-1H-imidazol-4-yl)benzoic acid
4-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}phenol
(2S)-2-{2-[1-(2-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamido}propanamide
3-(2-oxoazepan-1-yl)-N-[(1-phenylcyclopentyl)methyl]propanamide
4-({ethyl[(2-fluorophenyl)methyl]amino}methyl)-5-(hydroxymethyl)-2-methylpyridin-3-ol
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[4-(pyrrolidin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]propan-1-one
5-{3-[4-(3-methoxybenzoyl)piperazin-1-yl]-3-oxopropyl}imidazolidine-2,4-dione
1-benzyl-N,N-dimethyl-5-[methyl(thiophen-3-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(3,5-dimethylphenyl)-4-[4-(1H-pyrazol-1-yl)benzoyl]piperazin-2-one
7-{[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]methyl}-4-methyl-2H-chromen-2-one
2-[4-(1-phenylpiperidin-4-yl)-1-(propan-2-yl)piperazin-2-yl]ethan-1-ol
6-({2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}methyl)-1,4-oxazepan-6-ol
1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,5-dimethyl-1H-1,2,4-triazole
1-(cyclohexylmethyl)-3-hydroxy-3-(thiomorpholin-4-ylmethyl)piperidin-2-one
N-(1,3-benzoxazol-2-ylmethyl)-1-[(4-chlorophenyl)methyl]-N-methyl-6-oxopiperidine-3-carboxamide
2-ethoxy-N-[1-(4-fluorophenyl)-4-(morpholin-4-yl)-1H-indazol-3-yl]acetamide
1-{2-[benzyl(methyl)amino]acetyl}-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
3-(1-methylpiperidin-2-yl)-N-[2-(4-phenylpyrimidin-2-yl)ethyl]propanamide
1-(azepan-1-yl)-3-[2-methoxy-4-({[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
2-amino-1-[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
1-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-5,5-diphenylpiperidin-2-one
4-(2-methylpropyl)-6-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]pyrimidin-2-amine
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carboxamide
5-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-2,3-dimethyl-1H-indole
1-(4-{[cyclopropyl(pyridin-4-ylmethyl)amino]methyl}thiophen-2-yl)ethan-1-one
1-(1-methylpiperidin-4-yl)-4-[(1s,4s)-4-aminocyclohexyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-{[4-({[3-(trifluoromethyl)phenyl]methyl}amino)quinazolin-2-yl]methyl}benzenesulfonamide
N-methyl-5-propyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1,2-oxazole-3-carboxamide
4-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]benzonitrile
4-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-ylmethyl]-N-(1,3-dihydro-2-benzofuran-5-yl)benzamide
1-benzyl-8-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[N-cycloheptyl-1-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)formamido]acetic acid
N-{4-[4-(azepan-1-yl)butanamido]phenyl}pentanamide
3,3,3-trifluoro-N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}propanamide
3-[3-(4-phenylpiperazin-1-yl)piperidine-1-carbonyl]-1H-indole
N-methyl-1-(propan-2-yl)-N-[1-(1,3-thiazol-5-yl)ethyl]piperidine-4-carboxamide
1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-3-hydroxypropan-1-one
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
3-[({1-[6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidin-4-yl}oxy)methyl]pyridine
5-[2-(1,2-benzoxazol-3-yl)acetyl]-N-cyclopropyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
4-[3-(4-chlorophenyl)-5-[2-(1H-1,2,3,4-tetrazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl]-1-methylpiperidine
2-(1H-indol-3-yl)-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]acetamide
1-({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-phenyl-1,4-diazepane
2-(2-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydrophthalazin-1-one
6-[1-(pyridin-4-ylmethyl)-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-indole
2-(2-ethyl-1H-imidazol-1-yl)-N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]acetamide