提示: 按住Ctrl键可以同时选择多个官能团
2-{4-[3-(1,4-oxazepane-4-carbonyl)piperidin-1-yl]piperidin-1-yl}-1,3-benzoxazole
N-(1-{1-[(3-acetylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenylpropanamide
7-hydroxy-6-methyl-4-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-1,2,3,4-tetrahydroquinolin-2-one
methyl 3-benzamido-5-[(4-hydroxybutan-2-yl)amino]-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-{1-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-2-(2-fluorophenyl)ethyl}-N,2-dimethylfuran-3-carboxamide
N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-5-(oxolan-2-yl)thiophene-2-carboxamide
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]thiophene-2-carboxamide
1-{2-[(2-methylprop-2-en-1-yl)oxy]phenyl}-5-oxopyrrolidine-3-carboxylic acid
(1S,4S)-2-(4-chloro-2-methoxy-5-methylphenyl)-5-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-2,5-diazabicyclo[2.2.1]heptan-3-one
4-[1-benzyl-5-(3-phenyl-1,2-oxazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
5-(cyclohex-3-en-1-ylmethyl)-2-(4-methoxyphenyl)-6-methyl-2,3,4,5-tetrahydro-1,5-benzothiazepine
N-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-(1H-imidazol-2-yl)benzamide
3-(2-methoxyphenoxy)-1-[3-(methylsulfanyl)butyl]azetidine
1-methyl-4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N,1,3-trimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
6-{3-[(2H-1,3-benzodioxol-5-yl)amino]piperidin-1-yl}pyridine-2-carbonitrile
1-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
6-methoxy-1-methyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1H-indole-2-carboxamide
ethyl 4-benzyl-1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidine-4-carboxylate
N-ethyl-N-[1-(1-phenyl-1H-1,2,3-triazole-5-carbonyl)pyrrolidin-3-yl]acetamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(oxan-4-yl)pyrrolidine-3-carboxylic acid
2-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-yl]-N-[2-(4-methoxyphenyl)ethyl]acetamide
N-[2-(3-hydroxypiperidin-1-yl)ethyl]-2,6-dimethylquinoline-3-carboxamide
N,N-dimethyl-2-[(1S,5R)-3-{2-methylpyrido[2,3-d]pyrimidin-4-yl}-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
N-({1-[(3-acetylphenyl)methyl]pyrrolidin-3-yl}methyl)benzamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(1H-indazole-3-carbonyl)piperidin-3-amine
2-{5-[1-(3-cyclopentylpropanoyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetic acid
(3S,9aR)-2,3-dimethyl-8-(thiophen-3-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinoline
2-hydroxy-N-{2-[4-(pyridin-4-ylmethyl)morpholin-2-yl]ethyl}pyridine-3-carboxamide
1-[(3S,4R)-1-(2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
5-cyclopropyl-1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-3-(piperidin-3-yl)benzamide
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
2-{4-[(2,2-dimethylmorpholin-4-yl)methyl]phenyl}-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
N-[2-(4-chlorophenyl)-2-(pyrrolidin-1-yl)ethyl]-1H,4H,6H,7H-pyrano[4,3-c]pyrazole-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}propanamide
3-hydroxy-3-({[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-1-(3-phenylpropyl)piperidin-2-one
2-[4-({4-[(6-methylpyridin-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-ol
N-[(3R,4S)-4-cyclopropyl-1-(oxan-4-yl)pyrrolidin-3-yl]pyridine-4-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-amino-6-(3,5-dimethyl-1H-pyrazol-4-yl)-4-(4-hydroxy-2-methoxyphenyl)pyridine-3-carbonitrile
1-(2-methoxyethyl)-8-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{[1-(5-methylpyridine-3-carbonyl)pyrrolidin-3-yl]methyl}benzamide
2-(2-{[4-(2-amino-6-hydroxypyrimidin-4-yl)piperazin-1-yl]methyl}phenoxy)acetamide
(1S,6R)-9-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]acetamide
2-(2-{4-phenyl-5-[4-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}ethoxy)ethan-1-ol
N,5-dimethyl-4-[(pyridin-2-ylmethyl)amino]-N-[1-(thiophen-2-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
3-({[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}methyl)-1-(2,2-dimethylpropyl)-3-hydroxypiperidin-2-one