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2-(4-fluorophenoxy)-1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-4-(1,2,4-oxadiazol-3-yl)pyridine
2-(4-chloro-2-methylphenoxy)-1-[3-(4-fluorophenoxy)azetidin-1-yl]ethan-1-one
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
N-[(3S,4R)-1-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
5-(2-chlorophenyl)-N-ethyl-2-methyl-N-(oxan-4-ylmethyl)furan-3-carboxamide
1-(2-chloro-6-fluorobenzoyl)-3-[2-(4-fluorophenyl)ethyl]piperidine
N-(4-fluorophenyl)-1-(2-methyl-1-benzofuran-5-carbonyl)piperidin-3-amine
N-[1-(1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-2,2-dimethylpropanamide
1-{2-[2-(3-chlorophenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
1-{3-[3-(4-methoxyphenoxymethyl)piperidine-1-carbonyl]phenyl}ethan-1-one
8-(2,2-diphenylethyl)-1,3-dioxa-8-azaspiro[4.5]decan-2-one
[(2S)-1-{5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1H-pyrazole-3-carbonyl}pyrrolidin-2-yl]methanol
{[7-fluoro-2-(thiophen-3-yl)quinolin-3-yl]methyl}[(3,4,5-trimethoxyphenyl)methyl]amine
5-methyl-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]-1-propyl-1H-pyrazole-4-carboxamide
N-(1H-imidazol-2-ylmethyl)-N-methyl-1-(6-methyl-2-phenylpyrimidin-4-yl)piperidin-4-amine
(3E)-2-[4-(pyridin-4-yl)piperidin-1-yl]hept-3-enoic acid
2-[3-(3-fluorophenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-methyl-N-[3-(morpholin-4-yl)propyl]acetamide
(3S,4R)-1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-4-(3-methylthiophen-2-yl)piperidin-3-ol
1-methyl-3-propyl-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1H-pyrazole-5-carboxamide
8-(2,2-diphenylethyl)-1-ethyl-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-3-(N-methyl-1-{1-[1-(2-phenylethyl)piperidin-4-yl]piperidin-3-yl}formamido)propanamide
5-[3-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl](isoquinolin-5-ylmethyl)methylamine
[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl][1-(ethylsulfanyl)propan-2-yl]amine
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(2-methylbenzoyl)piperidine
N-(cyclopropylmethyl)-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(furan-2-ylmethyl)-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
1-(4-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-[(4-chlorophenyl)sulfanyl]ethan-1-one
propan-2-yl 2-chloro-5-[2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamido]benzoate
methyl 2-{4-[(2-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}piperidine-1-carboxylate
N-[(1S,2R)-2-aminocyclobutyl]-3-(4-chloro-1H-pyrazol-1-yl)propanamide
(2S,4R)-N-[(2-chloropyridin-3-yl)methyl]-4-(3-fluorobenzamido)-N-methylpyrrolidine-2-carboxamide
1-{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-methyl-1,4-diazepane
9-(morpholine-4-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-5-{4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}pyrazine
2-{1-[(1-cycloheptanecarbonylpiperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}pyridine
4-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-1-phenylpiperazin-2-one
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
(2S,4S)-4-amino-1-(2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}acetyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)quinoline-3-carboxamide
(4aR,7aS)-1-propanoyl-4-(pyridine-3-sulfonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-benzyl-1-cyclopropyl-4-oxo-5-(3-oxo-4-phenylpiperazine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N-(2-fluorophenyl)-5-[2-(pyridin-2-yl)-1H-imidazol-1-yl]furan-2-carboxamide
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(propan-2-yloxy)propan-1-one
N-[(3S,7S,8aS)-3-(1H-indol-3-ylmethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-phenylbenzamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-{pyrazolo[1,5-a]pyridine-3-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-methyl-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
1-[(4-methanesulfonylphenyl)methyl]-3-(1-methyl-1H-imidazol-2-yl)piperidine
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-N,N-dimethylpiperidine-1-sulfonamide