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(2S)-2-[2-(2-ethoxyphenyl)-1H-imidazol-1-yl]-4-(methylsulfanyl)butan-1-ol
2-(4-{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)ethan-1-ol
3-(4-ethyl-1H-pyrazol-5-yl)-1-[5-(propan-2-yl)-1,3-oxazole-4-carbonyl]piperidine
6-(2-aminoethyl)-2-(3-{[methyl(1H-pyrazol-5-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
3-hexyl-8-(2-methyl-1,3-thiazole-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[2-(2-ethoxyphenyl)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-3-cyclohexyl-1H-pyrazole-4-carboxamide
6-(aminomethyl)-2-(2-methyl-1,3-thiazol-4-yl)-3,4-dihydropyrimidin-4-one
2-{1-[(3-methoxyphenyl)methyl]-4-(quinolin-6-ylmethyl)piperazin-2-yl}ethan-1-ol
N-ethyl-N-(1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)acetamide
N-(2,3-dihydro-1H-inden-1-yl)-2-(dimethylamino)-2,3-dihydro-1H-indene-2-carboxamide
1-[5-(2-chloro-4-fluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-3-(methoxymethyl)piperidine
2-(2-methoxyphenoxy)-N-({1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-yl}methyl)acetamide
5-chloro-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N-methylpyridine-2-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4-(5-methylfuran-2-yl)benzamide
3-(1-cyclopentylpiperidin-3-yl)-N-[(5-methylfuran-2-yl)methyl]propanamide
N-[(2,3-difluorophenyl)methyl]-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(1S,5R)-6-(cyclopropanesulfonyl)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
4-[(diethylamino)methyl]-5-ethyl-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methylfuran-2-carboxamide
1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-4-[(3-fluorophenyl)methyl]piperazine
2-(1-{1-[(5-ethylpyridin-2-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}butanamide
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-N,2,7-trimethylimidazo[1,2-a]pyridine-3-carboxamide
1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-4-[1-(2,2-dimethylpropyl)pyrrolidin-3-yl]piperidine
N-ethyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
2-{1-[(2-methylphenyl)methyl]-4-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}piperazin-2-yl}ethan-1-ol
3-({[(2-aminopyrimidin-5-yl)methyl](methyl)amino}methyl)-3-hydroxy-1-(2-phenylethyl)piperidin-2-one
1-(2-{pyrazolo[1,5-a]pyridin-7-yl}pyrimidin-4-yl)piperidin-3-ol
N-[(2R,3R)-1'-[(4-fluoro-3-methoxyphenyl)methyl]-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxybenzamide
1-[2-(1H-imidazol-2-yl)benzoyl]-3-(3-methoxypropyl)piperidine-3-carboxylic acid
7-ethyl-2-(3-ethyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-({1-ethyl-5-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-3-yl}methyl)-1-methylpiperidine
2-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]-N-[2-(4-methoxyphenyl)ethyl]acetamide
4-({2-[3-(dimethylamino)-2-hydroxypropoxy]-5-methoxyphenyl}methyl)-1-methylpiperazin-2-one
methyl (2S,4R)-1-[(2E)-3-(5-chloro-2-hydroxyphenyl)-2-methylprop-2-en-1-yl]-4-(dimethylamino)pyrrolidine-2-carboxylate
N-[(1R,2S)-2-(methoxymethyl)cyclopentyl]-2,3,6-trimethylquinoline-4-carboxamide
2-[2-(2-hydroxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]-N-(1-methyl-1H-pyrazol-3-yl)acetamide
N-[(3-methoxyphenyl)methyl]-3-[1-(oxane-4-carbonyl)piperidin-3-yl]propanamide
4-methyl-1-{2-oxo-2-[4-(pyridin-4-yl)piperidin-1-yl]ethyl}-1,2-dihydroquinolin-2-one
(2S,4S)-4-amino-1-(2-methoxy-5-sulfamoylbenzoyl)pyrrolidine-2-carboxylic acid
4-(1H-1,3-benzodiazol-1-yl)-1-(furan-2-carbonyl)piperidine-4-carboxylic acid
1-({4-methyl-5-[1-(4-methylpent-3-en-1-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
(1S,5R)-3-(2,1,3-benzoxadiazol-4-ylmethyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{1-[(2-aminopyridin-3-yl)methyl]piperidin-3-yl}propanamide
N-methyl-N-{2-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]ethyl}methanesulfonamide
4-({4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
3-[(7-chloro-1-methyl-1H-indol-2-yl)formamido]-N-cyclohexylpropanamide
1-{2-[(2-ethoxyphenyl)carbamoyl]acetyl}-N-ethylpyrrolidine-3-carboxamide
2-{2-amino-6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}-N-tert-butylbenzene-1-sulfonamide
2-{[3-(furan-2-yl)phenyl]methyl}-octahydropyrrolo[1,2-a]piperazine