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4-ethyl-3-({1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-4-yl}methyl)-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
7-(5-chloropyridin-2-yl)-4-(2,2-dimethylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperidin-4-yl)(pyridin-2-yl)methanol
1'-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
3-(4-{3-[(1R,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]pyridin-2-yl}phenyl)propanoic acid
4-chloro-2-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidine-1-carbonyl]phenol
4-[5-(5-propyl-1,2-oxazol-3-yl)-1,2,4-oxadiazol-3-yl]pyridine
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-4-(4-methylpiperazin-1-yl)benzamide
N-[2-(5-methylfuran-2-yl)ethyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-3-(thiophen-3-yl)-1H-pyrazole-5-carboxamide
(1R,7S)-3-(2,2-dimethylpropyl)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
4-fluoro-N-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}benzamide
methyl 3-[1-(4-chlorophenyl)cyclopropaneamido]-5-{[2-(3-fluorophenyl)acetamido]methyl}benzoate
2-(6-chloro-2H-1,3-benzodioxol-5-yl)-7-methyl-1H-1,3-benzodiazole
(1R,9S)-5-amino-3-(6-methoxy-2H-1,3-benzodioxol-5-yl)-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
2-cyclopropyl-8-[2-(1H-imidazol-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
(3R)-1-{4-[4-(2-chlorophenyl)piperidin-4-yl]pyrimidin-2-yl}pyrrolidin-3-ol
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
2-(5-{6-chloroimidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-3-yl)pyrazine
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-4-(2-oxopyrrolidin-1-yl)butanamide
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-3-{[(3-methylthiophen-2-yl)methyl]amino}benzamide
3-(1H-1,3-benzodiazol-1-yl)-1-[3-(2-methoxybenzoyl)piperidin-1-yl]propan-1-one
(1R,5R)-3-methanesulfonyl-6-[5-(methoxymethyl)furan-2-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
2,3,4-trimethoxy-N-({5-[4-(methylsulfanyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)benzamide
3,3-diethyl-1-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-3-yl)phenyl]urea
6,6-dimethyl-1-(2-methylphenyl)-N-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
[7-(5-fluoro-3,8-dimethylquinolin-2-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methanamine
3-[1-(1,1-dioxo-1λ6-thian-4-yl)piperidin-4-yl]-1-(2-hydroxypyridin-3-yl)urea
1-(3-{[(4-carbamoyl-3-chlorophenyl)carbamoyl]amino}propyl)piperidine-3-carboxamide
N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-1H-1,3-benzodiazole-5-carboxamide
2-amino-6-(furan-2-yl)-4-[5-(oxolan-2-yl)thiophen-2-yl]pyridine-3-carbonitrile
2-(5-{3,9-diazaspiro[5.5]undecane-3-carbonyl}-1H-pyrazol-3-yl)phenol
N,N-dimethyl-5-{[8-(2-methylquinolin-4-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}pyrimidin-2-amine
(3R,4S)-4-propyl-1-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]pyrrolidin-3-amine
4-(2,4-dioxoimidazolidin-1-yl)-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]benzamide
1-(3-{3-oxo-3-[4-(pyridin-2-yl)piperazin-1-yl]propyl}piperidin-1-yl)propane-1,2-dione
3-(1-methyl-1H-imidazol-2-yl)-1-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]piperidine
2-{3-[4-(dimethylamino)azepan-1-yl]-3-oxopropyl}-2,3-dihydro-1H-isoindol-1-one
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
1-cyclohexyl-5-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
2-{[4-(2-aminopyridin-4-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}acetic acid
2-[(4aR,8aR)-4a-hydroxy-7-methanesulfonyl-decahydro-2,7-naphthyridin-2-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-[5-(1H-imidazol-4-ylmethyl)-3-phenyl-1H-1,2,4-triazol-1-yl]pyridine
1-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
methyl({[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl})(3-phenylpropyl)amine
4-benzyl-3-ethyl-1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1,4-diazepan-5-one
N-cyclopropyl-5-(2-oxo-1,2,3,4-tetrahydroquinoline-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-[(3-fluorophenyl)methyl]-5-[4-(2-methoxyethyl)piperazine-1-carbonyl]piperidin-2-one
2-{5-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1H-pyrazol-3-yl}pyridine