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(2S,4R)-4-amino-1-(3-methoxybenzenesulfonyl)-N-methylpyrrolidine-2-carboxamide
methyl 1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-4-carboxylate
1-methyl-N-(oxolan-2-ylmethyl)-N-propyl-1H-indole-2-carboxamide
(8R,9aS)-8-hydroxy-2-[3-(1H-imidazol-1-yl)propyl]-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]benzamide
N-[(1R,3S)-3-[(2,3-dihydro-1H-inden-2-yl)carbamoyl]cyclopentyl]-1-propyl-1H-pyrazole-5-carboxamide
N-benzyl-2-[3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]acetamide
3-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-4-yl}-1-(4-phenylpiperazin-1-yl)propan-1-one
1-(4-fluorobenzoyl)-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
2-(6-{6-[(piperidin-4-yl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-3-yl)acetic acid
1-(2,1,3-benzoxadiazol-5-ylmethyl)-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}pyridine
1-[(4-methoxyphenyl)methyl]-4-(2-methyl-1,3-thiazole-4-carbonyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
1-(4-{[5-(hydroxymethyl)furan-2-yl]methyl}-1,4-diazepan-1-yl)-2-methoxyethan-1-one
methyl 2-[(3,4-difluorophenyl)sulfamoyl]-6-(2,2-dimethylpropanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-[3-phenyl-5-(1,2,5-trimethyl-1H-pyrrol-3-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
(4aR,7aS)-1-methyl-4-[2-methyl-2-(3-methylphenoxy)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(4-{[(3-chlorophenyl)methyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)({[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
4-(1H-imidazol-2-yl)-1-[2-(1H-imidazol-4-yl)ethyl]-1H-1,2,3-triazole
1-cyclopropanecarbonyl-N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]piperidine-4-carboxamide
(3S,5R)-1-[(3-ethyl-1H-pyrazol-5-yl)methyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
2-(furan-3-yl)-4-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazole
1-(2-methoxyphenyl)-3-(1-{1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
1'-[2-(ethylamino)pyrimidine-5-carbonyl]-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
N-[2-(2-fluorophenyl)-1-[1-(quinoxalin-5-ylmethyl)piperidin-4-yl]ethyl]-N-methylthiophene-3-carboxamide
3-phenyl-1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)prop-2-yn-1-one
3-cyclobutyl-4-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-[(4-benzylpiperidin-1-yl)methyl]-N-[(2S)-1-hydroxy-3,3-dimethylbutan-2-yl]-1,2-oxazole-3-carboxamide
N-cyclohexyl-3-[2-(2,3,6-trimethylphenoxy)acetamido]propanamide
[(4aS,8aR)-6-(oxan-4-yl)-1-(1H-1,2,4-triazole-5-carbonyl)-decahydro-1,6-naphthyridin-4a-yl]methanol
4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-N,N-diethylbenzamide
[(2S,4R)-1-{2-[cyclohexyl(methyl)amino]pyridine-3-carbonyl}-4-(dimethylamino)pyrrolidin-2-yl]methanol
1-[(3S,4S)-3-hydroxy-4-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]-2-(2,3,4-trifluorophenyl)ethan-1-one
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-6-methoxyhexan-1-one
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
5-{[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]methyl}-N-(propan-2-yl)pyrimidin-2-amine
(3S,4R)-1-[2-methyl-2-(morpholin-4-yl)propyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
2-methanesulfonyl-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
4-(naphthalen-2-ylmethyl)-3-{2-oxo-2-[4-(pyrrolidin-1-yl)piperidin-1-yl]ethyl}piperazin-2-one
2-{1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]pyrrolidin-2-yl}-1,3-benzothiazole
2-(4-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)-1,3-benzothiazole
(1R,5S,8S)-3-[(2,3,4-trifluorophenyl)methyl]-3-azabicyclo[3.2.1]octan-8-ol
2-(3-fluorophenyl)-1-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
4-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
3-hydroxy-1-[(3-methylphenyl)methyl]-3-(1,2-oxazolidin-2-ylmethyl)piperidin-2-one
N-{1-[1-(1-carbamoylethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxybenzamide
6-(but-3-enoyl)-N-[4-(methylsulfanyl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
2-(3-chlorophenyl)-2-hydroxy-N-(isoquinolin-5-ylmethyl)-N-methylacetamide
1-(6-cyanopyridine-3-carbonyl)-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide