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(1r,4r)-4-methyl-N-{2-[4-(pyridin-4-ylmethyl)morpholin-2-yl]ethyl}cyclohexane-1-carboxamide
4-({1-[1-(propan-2-yl)piperidine-4-carbonyl]azetidin-3-yl}oxy)benzoic acid
2-(2-methoxy-5-methylphenyl)-2-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]acetic acid
(4S)-1-(4-hydroxy-3-methylbenzoyl)-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
methyl (2S,4R)-4-(2-cyclopropylquinoline-4-amido)-1-[(2-methoxyphenyl)methyl]pyrrolidine-2-carboxylate
[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
[(2-methoxyphenyl)methyl](2-phenylethyl)(pyridin-3-ylmethyl)amine
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetamide
(3R,4R)-1-[(2-fluoro-5-methoxyphenyl)methyl]-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
3-{1-[3-(methylsulfanyl)propanoyl]piperidin-3-yl}-N-[4-(trifluoromethyl)phenyl]propanamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]propanamide
N-(3-acetamidophenyl)-4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carboxamide
N-cyclopropyl-2-methyl-N-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}propanamide
2-methoxy-N-{1-[1-(quinolin-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N-{[3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(1,2-oxazinan-2-yl)propanamide
[3-(cyclopropylmethyl)-1-[(5-ethylpyridin-2-yl)methyl]piperidin-3-yl]methanol
4-(1H-imidazol-2-yl)-1-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H-1,2,3-triazole
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(3-methylphenoxymethyl)piperidine
2-(5,6,7,8-tetrahydronaphthalen-2-yloxy)-N-[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]butanamide
1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-4-(1,2,4-oxadiazol-3-yl)piperidine
N-({1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[(4-hydroxy-1-methylpiperidin-4-yl)methyl]-1H-pyrazole-3-carboxamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-[(3-methoxyphenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(3-{8-methyl-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}phenyl)imidazolidin-2-one
{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}(methyl)[(5-methylfuran-2-yl)methyl]amine
1-[(2-{3-[cyclohexyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]piperidine-4-carbonitrile
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}acetamide
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
2-{4-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]piperazin-1-yl}pyridine-3-carbonitrile
(4aR,8aR)-2-cyclobutanecarbonyl-7-[(2,5-dimethylphenyl)methyl]-decahydro-2,7-naphthyridin-4a-ol
5-{[3-(naphthalene-1-carbonyl)piperidin-1-yl]methyl}-2,1,3-benzoxadiazole
3-cyclopropaneamido-N-[2-(ethanesulfonyl)ethyl]-4-methylbenzamide
N-{1-[7-(pyrazin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]pyrrolidin-3-yl}acetamide
1-(2-fluorophenyl)-3-methyl-5-[1-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
N-[(1R,2R)-1-[(7-fluoroquinazolin-4-yl)amino]-2,3-dihydro-1H-inden-2-yl]acetamide
N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
[1-(1-{[1-(3-chlorophenyl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methanamine
7-methyl-3-(quinolin-2-ylmethyl)-3,7,11-triazaspiro[5.6]dodecan-12-one
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(4-methylbenzoyl)piperidin-4-yl]oxy}benzamide
9-(1-ethyl-1H-pyrazole-5-carbonyl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(1-methyl-1H-indol-3-yl)ethan-1-one
5-hydroxy-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}pyridine-2-carboxamide
2-(2,2-dimethyloxan-4-yl)-1-(2-phenoxyethyl)-1H-imidazole
4-{1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]pyrrolidin-2-yl}-3,5-dimethyl-1,2-oxazole
3-(2-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-oxoethyl)-3,4-dihydroquinazolin-4-one
2-(adamantan-1-yl)-N-[2-hydroxy-2-(1-methyl-1H-imidazol-2-yl)ethyl]acetamide
3-(4-chlorobenzoyl)-1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]piperidine
6-{[(2R)-2-carbamoylpyrrolidin-1-yl]methyl}-2-oxo-N-(quinolin-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
4-chloro-2-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1H-indole
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)-2-(morpholin-4-yl)pyridine-3-carboxamide