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2-ethoxy-N-[(3R,4S)-4-(propan-2-yl)-1-(3,3,3-trifluoropropyl)pyrrolidin-3-yl]acetamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(2-fluorobenzoyl)piperidin-3-ol
2-[(2-phenylpyrimidin-5-yl)methyl]-2,8-diazaspiro[4.5]decane
6-[(3R,4S)-3-(3-ethoxypropanamido)-4-(propan-2-yl)pyrrolidin-1-yl]pyrazine-2-carboxamide
N-[(2S)-1-{3-[5-(4-fluorophenyl)-2-methylpyrimidin-4-yl]piperidin-1-yl}-1-oxopropan-2-yl]acetamide
3-(dimethylamino)-N-(2-methyl-1-benzofuran-7-yl)pyrrolidine-1-carboxamide
methyl (2S,4R)-4-hydroxy-1-{[5-(pyrimidin-2-ylsulfanyl)furan-2-yl]methyl}pyrrolidine-2-carboxylate
3-(methanesulfonylmethyl)-1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperidine
N-[4-methoxy-2-(2-methylpropanamido)phenyl]-1,2,3-thiadiazole-4-carboxamide
1-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-3-(1-ethyl-3-methyl-1H-pyrazol-4-yl)urea
1-(6-methyl-3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}quinolin-2-yl)piperidin-3-ol
2-methyl-8-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
2-{1-[(4-fluorophenyl)methyl]-4-[5-(propan-2-yl)pyrimidin-4-yl]piperazin-2-yl}ethan-1-ol
N-(2-methoxyethyl)-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]-N-(propan-2-yl)acetamide
2-(2-{4-[(dimethylamino)methyl]phenyl}pyrrolidin-1-yl)-2-oxoacetamide
1-{1-[2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]azetidin-3-yl}-2-methylpiperidine
N-methyl-2-[(2-methyl-5-propylpyrimidin-4-yl)amino]ethane-1-sulfonamide
1-[(3R,4R)-4-cyclopropyl-4-hydroxy-3-methylpiperidin-1-yl]-2-(pyrrolidin-1-yl)ethan-1-one
1-{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-ethylpiperazine
2-(3-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}phenoxymethyl)pyridine
2-[(2-butoxy-3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
(3S,4R)-4-methyl-1-{7-methyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}piperidine-3,4-diol
7-(cyclopropylmethyl)-6-(2-fluoro-4-methoxyphenyl)-2-(3-hydroxyazetidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
1-[2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]-2-(thiophen-3-yl)ethan-1-one
1'-[5-(methoxymethyl)thiophene-2-carbonyl]-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]ethan-1-one
6,8-dimethyl-3-{1-[2-(1H-pyrazol-4-yl)ethyl]-1H-imidazol-2-yl}-1,2-dihydroquinolin-2-one
3-(1H-imidazol-2-yl)-1-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]piperidine
2-(2-methylpropyl)-8-[2-(oxan-2-ylmethoxy)acetyl]-2,8-diazaspiro[4.5]decan-3-one
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-3-(4-methoxy-2-methylbenzoyl)piperidine
8-[3-(6-oxo-1,6-dihydropyridazin-3-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-(2-methylpiperidin-1-yl)-2-oxo-N-(prop-2-en-1-yl)-N-(propan-2-yl)acetamide
N-{[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-3-yl]methyl}-3,5-dimethoxybenzamide
(3-phenylprop-2-yn-1-yl)(propyl){[6-(trifluoromethyl)pyridin-3-yl]methyl}amine
4-{[(2,3-dimethoxyphenyl)methyl]amino}-5-methyl-N-[2-(methylsulfanyl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
5-methyl-4-{2-[methyl(pyridin-2-ylmethyl)amino]acetyl}-1-(2-methylphenyl)piperazin-2-one
1-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(thiophen-2-yl)propan-1-one
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
N,5-dimethyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}-1,3,4-oxadiazol-2-amine
2-(2-methyl-1,3-thiazol-4-yl)-1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
3-methyl-8-[2-(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2S)-2-{4-oxo-3H,4H-thieno[3,2-d]pyrimidin-3-yl}-3-phenylpropanamide
7-(3-chlorophenyl)-4-[(1-methyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[2-(3-fluorophenyl)ethyl]-1-methanesulfonylpiperidine
1-(5-chloropyridin-2-yl)-4-{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperazine
3-(2-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}-2-oxoethyl)-3,4-dihydroquinazolin-4-one
[(3R,4S)-1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
(3S,4S)-1-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
3-(2-methyl-1H-imidazol-1-yl)-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
4-(4-methyl-1H-pyrazol-1-yl)-1-(quinolin-8-ylmethyl)piperidine-4-carboxylic acid