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N-[3-(morpholin-4-yl)propyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
3-fluoro-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}pyridin-2-amine
2-ethyl-5-[2-(morpholin-4-ylmethyl)phenyl]-1,3-benzoxazole
6-methyl-N-[(1-methylpyrrolidin-3-yl)methyl]-1-(propan-2-yl)-1H-pyrazolo[3,4-b]pyridine-4-carboxamide
(3R,5S)-1-[(4-hydroxyphenyl)methyl]-N-(3-methoxypropyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
2-(2-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}phenoxy)ethan-1-ol
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5-(2,5-dimethylphenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
N-(2,3-dimethylphenyl)-4-methyl-1,2,3,6-tetrahydropyridine-1-carboxamide
3-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-3H,4H-pyrido[4,3-d]pyrimidin-4-one
(1S,5R)-6-(2H-1,3-benzodioxole-5-carbonyl)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane
methyl 3-[1-(4-chlorophenyl)cyclopropaneamido]-5-[(cyclobutylformamido)methyl]benzoate
(3S,4R)-4-(hydroxymethyl)-1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}piperidin-3-ol
N-{[6,7-dimethoxy-2-(3-methoxyphenyl)quinolin-3-yl]methyl}-5,6-dimethyl-2-oxo-N-(oxolan-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
1-(2-fluoroethyl)-5-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-4-phenyl-1H-imidazole
(3S,4S)-1-[2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}[(2-methylpyrimidin-5-yl)methyl]amine
1-{1-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-[(3-fluorophenyl)methyl]-4-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperazine
4-[(3-methyl-1H-pyrazol-5-yl)methyl]-3-propylmorpholine
N-(3-chloro-4-methoxyphenyl)-3-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]propanamide
N-[(1R,3R)-3-aminocyclopentyl]-4-methoxy-2,3,6-trimethylbenzene-1-sulfonamide
2-(3-phenylpiperidin-1-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}acetamide
(2S,4S)-4-(4-cyanooxane-4-amido)-N-ethyl-1-(1H-imidazol-2-ylmethyl)pyrrolidine-2-carboxamide
3-methoxy-1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
6-methyl-1-[1-oxo-1-(pyrrolidin-1-yl)propan-2-yl]-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
2-methyl-4-{3-[4-(2,2,2-trifluoroethyl)piperazine-1-carbonyl]phenyl}butan-2-ol
N-(5-chloro-2-methoxyphenyl)-3-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-3-yl]propanamide
(2S,4R)-N,N-diethyl-1-(2-fluoro-4-methylbenzoyl)-4-(2-hydroxyacetamido)pyrrolidine-2-carboxamide
1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(thiophen-2-yl)ethan-1-one
2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[4-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]ethan-1-one
1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(2,2,2-trifluoroethyl)piperazine
2-({6-[3-(1H-pyrazol-5-yl)piperidin-1-yl]pyrimidin-4-yl}amino)ethan-1-ol
N,1-dimethyl-N-(1,2-oxazol-3-ylmethyl)-3-propyl-1H-pyrazole-5-carboxamide
4-(1,3-benzoxazol-2-yl)-N-(4-ethoxyphenyl)piperazine-1-carboxamide
(3aR,6aS)-2-ethyl-5-(morpholine-4-sulfonyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-methyl-5-[({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]pyrrolidin-2-one
N-(2,2-dimethylpropyl)-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
1-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-3-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}urea
3-hydroxy-S-[2-(3-methylbutanoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]butane-1-sulfonamido
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
1-(1-{2-[(2-chlorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-4-carbonyl)piperidine-3-carboxamide
5-{1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
9-[(4-methoxyphenyl)methyl]-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-ethyl-5-{[5-(4-methoxyphenyl)furan-2-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
8-[2-(benzyloxy)acetyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-3-(propan-2-yl)-1,2-oxazole
2-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]-1,2,3,4-tetrahydroisoquinoline
methyl 4-[(4-{2-[(2-chlorophenyl)carbamoyl]ethyl}piperidin-1-yl)methyl]benzoate
1-(2-methoxyacetyl)-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}piperidine-3-carboxamide
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methyl-1,4-diazepan-5-one