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1-[(5-ethylfuran-2-yl)methyl]-4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazine
(2S,4S)-4-amino-1-{[(2-fluorophenyl)carbamoyl]carbonyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-[5-(6-phenylpyridazin-3-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
7-(4-chlorophenyl)-2-(dimethyl-1,2-oxazol-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5-(azepane-1-carbonyl)-1-(butan-2-yl)-N-[2-methyl-2-(morpholin-4-yl)propyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
1-[(2,5-difluorophenyl)methyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
(3aS,6aR)-3-cyclopentyl-5-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-[(dimethylamino)methyl]-1-[(6-methoxy-2H-chromen-3-yl)methyl]piperidin-3-ol
1-[(2-chloro-4-fluorophenyl)methyl]-N-[1-(thiophen-2-yl)propan-2-yl]-1H-1,2,3-triazole-4-carboxamide
3-[(3-methyloxetan-3-yl)methyl]-1-(2-{[(4-methylphenyl)methyl]sulfanyl}phenyl)urea
(3R,9aR)-8-[(3-methylphenyl)methyl]-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-{[2-(1-methyl-1H-pyrazol-5-yl)ethyl]sulfamoyl}-N-[(2S)-oxolan-2-ylmethyl]benzamide
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-ethyl-6-methyl-4-oxo-1-[2-(piperidin-1-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
6-[2-(2-carboxyethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]-5-chloropyridine-3-carboxylic acid
3-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-5-(2-methylpropyl)-1,2,4-oxadiazole
2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decane
5-[3-(furan-2-yl)-3-phenylpropanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
6-methyl-N-{3-[(pyridin-3-yl)amino]propyl}imidazo[1,2-a]pyridine-2-carboxamide
4-(2-oxo-2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
2-{1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-1-oxobutan-2-yl}-2,3-dihydro-1H-isoindol-1-one
methyl 2-{8-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
2-(4-tert-butylphenoxymethyl)-4-hydroxy-N-(2-methanesulfonylethyl)pyrimidine-5-carboxamide
1-{[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}-4-phenylpyrrolidin-2-one
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
N-{[3-(cyclopentyloxy)phenyl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)-N-[(3S)-2-oxoazepan-3-yl]propanamide
3-{1-[2-(3-chloro-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]piperidin-4-yl}-N-(3-methylphenyl)propanamide
3-(pyrazin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[4-(4-{[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]amino}piperidin-1-yl)phenyl]pyrazine-2-carboxamide
4-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}methyl)-1H-pyrazole-3-carboxylic acid
(2R,3R)-1'-[(5-hydroxy-2-methoxyphenyl)methyl]-3-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-tert-butyl-3-oxo-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-{[6-(4-cyanophenyl)pyridin-3-yl]methyl}acetamide
2-{4-[(2,5-difluorophenyl)methyl]-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
7-(cyclohexylmethyl)-2-(pyridine-3-sulfonyl)-2,7-diazaspiro[4.5]decan-6-one
1-methanesulfonyl-4-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperazine
N,2,7-trimethyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)quinoline-4-carboxamide
1-[4-(6-cyclopropylpyrimidin-4-yl)-1,4-diazepan-1-yl]-2-methoxyethan-1-one
N-[(3,4-difluorophenyl)methyl]-2,6-dimethylpyridine-4-carboxamide
1-[2-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-oxoethyl]-3,3-dimethylurea
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
1-[6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidin-4-ol
N-[3-(pyrrolidine-1-carbonyl)-5-[({[3-(trifluoromethyl)phenyl]methyl}amino)methyl]phenyl]pyridine-2-carboxamide
(3R,7S,8aS)-7-({[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)-3-methyl-octahydropyrrolo[1,2-a]piperazine-1,4-dione
6-amino-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}pyridine-3-carboxamide
(1S,5R)-6-(3,5-difluoropyridine-2-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
1-(2-methylpyridin-4-yl)-4-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-1,4-diazepane
4-[(2-chloro-5-ethoxy-4-methoxyphenyl)methyl]-2-(trifluoromethyl)morpholine
N-(cyclohexylmethyl)-1-{1,3-dioxo-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
8-fluoro-2-[({3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}amino)methyl]quinolin-4-ol
N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide