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1-{[1-(cyclohexylmethyl)-2-methanesulfonyl-1H-imidazol-5-yl]methyl}-4-(pyrrolidin-1-yl)piperidine
1-{2-methylthieno[2,3-d]pyrimidin-4-yl}-4-[2-(pyrrolidin-1-yl)ethyl]piperidine
2-methyl-4-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidine-1-carbonyl}phenol
3-hydroxy-3-({[(5-methylfuran-2-yl)methyl]amino}methyl)-1-(3-phenylpropyl)piperidin-2-one
[4-(2-propyl-1,3-thiazole-4-carbonyl)-1,4-oxazepan-6-yl]methanol
4-{[5-(3-chlorothiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-methylpiperidine
2-(2,3-dimethylphenoxy)-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)acetamide
N'-(adamantan-1-yl)-N-[3-(1H-imidazol-1-yl)propyl]propanediamide
1-methyl-4-(2-methyl-1-benzofuran-7-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
(1S,6R)-3-{2-[4-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
1-[2,3-dimethyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}urea
6-butyl-2-(3-{[(2-hydroxyethyl)(methyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-6-methyl-4-oxo-4H-pyran-2-carboxamide
8-[2-(2-hydroxyethoxy)ethyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-methoxy-6-{4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyrimidin-2-amine
6-[4-(4-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-9H-purine
8-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}quinoline
2-(ethanesulfonyl)-5-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1-(3-phenylpropyl)-1H-imidazole
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]acetamide
2-(2-{[methyl(oxan-4-yl)amino]methyl}-4-(pyrimidin-2-yl)phenoxy)acetic acid
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
N,N-dimethyl-7-(propane-1-sulfonyl)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-chloro-N-{[1-(morpholin-4-ylmethyl)cyclopropyl]methyl}-5-(1H-pyrazol-1-yl)benzamide
(1R,7S)-3-(3,4-dimethylphenyl)-N-methyl-4-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
5-[1-(2-fluorophenyl)cyclopropyl]-3-(2-methoxyethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
1-[5-({8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)imidazo[2,1-b][1,3]thiazole-6-carbonyl]piperidine
4-(2-{3-[(2-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}ethyl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
5-(hydroxymethyl)-2-methyl-4-{[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]methyl}pyridin-3-ol
2-[(4-chlorophenyl)methyl]-8-[(4-methyl-1,3-thiazol-5-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-acetyl-8-[(2-aminopyrimidin-5-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5,6-dimethoxy-2-(oxan-2-ylmethyl)-1,2-dihydroisoquinolin-1-one
4-hydroxy-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
5-[2-(2-methoxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carbonyl]-1-methyl-1H-pyrrole-3-carbonitrile
4-[(2-methylpyridin-3-yl)oxy]-N,N-bis(prop-2-en-1-yl)piperidine-4-carboxamide
2-methyl-6-[(3-{3-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]phenyl}-1H-pyrazol-1-yl)methyl]pyridine
6-ethoxy-3-({ethyl[(3S,4R)-4-hydroxyoxolan-3-yl]amino}methyl)-1,2-dihydroquinolin-2-one
2-[(3,4-dimethoxyphenyl)methyl]-N-[2-(pyridin-2-yl)ethyl]-1,3-benzoxazole-6-carboxamide
2-chloro-N-[2-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
5-benzyl-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
6-[(2,2-dimethylmorpholin-4-yl)methyl]pyridine-2-carboxylic acid
N-methyl-1-[3-(morpholin-4-yl)propyl]-6-oxo-N-(1H-pyrazol-3-ylmethyl)piperidine-3-carboxamide
2-{4-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidine-1-carbonyl}morpholine
3-[(1H-imidazol-2-ylmethyl)sulfamoyl]-N-(oxan-4-ylmethyl)benzamide
5-({[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}carbamoyl)-1H-imidazole-4-carboxylic acid
1-[(2,4-difluorophenyl)methyl]-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)quinoxaline-6-carboxamide
1-(2,3-dimethyl-1H-indole-7-carbonyl)-4-[(2-fluorophenyl)methyl]-1,4-diazepan-5-one
(1R,5R)-N,N-dimethyl-6-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-[3-(1H-imidazol-1-yl)propyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(1S,6R)-9-(1-ethenyl-1H-pyrazole-4-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one