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N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyrazolo[1,5-a]pyridine-7-carboxamide
5-methyl-3-[1-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)pyrrolidin-2-yl]-1,2-oxazole
3-(2H-1,3-benzodioxol-5-yl)-5-{[3-(2-chlorophenyl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazole
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(4-methylphenyl)propan-1-one
5-[(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)methyl]-3-[(methylsulfanyl)methyl]-1,2,4-oxadiazole
N-{1-[1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methylbenzamide
5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-methyl-N-(pyrimidin-4-ylmethyl)pyridin-2-amine
5-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane-11-carbonyl}-N-ethylpyrimidin-2-amine
4-cyano-N,1-dimethyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrrole-2-carboxamide
3-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidine-1-carbonyl]benzonitrile
N-[(3S,4R)-1-[2-(4-chlorophenoxy)ethyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
1-[2-(3-fluorophenyl)ethyl]-6-oxo-N-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
(2-{[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl](thiophen-3-ylmethyl)amino}ethyl)dimethylamine
2-[3-(ethoxymethyl)-5-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]-4-methylpyridine
3-[2-(2,3-dihydro-1H-indol-1-yl)-2-oxoethyl]-1,3-diazinane-2,4-dione
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}but-2-ynamide
3-methyl-3-phenyl-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
8-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3S,9aR)-3-(cyclohexylmethyl)-8-(thiophen-3-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(4-fluoro-2-{[1,2,4]triazolo[4,3-a]pyrazin-3-yl}phenyl)-1H-pyrazole
2-[(3R,4R)-4-cyclopropyl-4-hydroxy-3-methylpiperidin-1-yl]-N-[2-(4-methoxyphenyl)ethyl]acetamide
(2R)-2-amino-N-{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}-4-methylpentanamide
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
2-methyl-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1-benzofuran-5-carboxamide
(3S,5R,9R)-11-[(3,4-dimethylphenyl)methyl]-5-hydroxy-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
1-ethyl-N-methyl-3-(thiomorpholine-4-carbonyl)-N-(thiophen-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(3-ethylphenyl)-2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-({4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)naphthalen-2-ol
1-[1-(pentan-2-yl)-1H-pyrazol-5-yl]-3-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}urea
1-[2-(diethylamino)acetyl]-N-[3-(4-fluorophenyl)phenyl]piperidine-3-carboxamide
3-ethyl-5-{[2-(2-phenylethynyl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-(5-fluoro-2-methylphenyl)acetamide
1-(3-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-sulfonyl}benzoyl)piperidine
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(4-methoxyphenyl)methyl]acetamide
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]ethan-1-one
2-[4-({[(4-ethyl-1,3-thiazol-2-yl)methyl]amino}methyl)phenoxy]-1-(morpholin-4-yl)ethan-1-one
1-{2-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
(3S,4R)-1-(4-fluoro-3-methylbenzoyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
7-(5-chloropyridin-2-yl)-4-(6-ethylpyrimidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-methyl-3-oxo-N-(2-oxoazepan-3-yl)-3,4-dihydroquinoxaline-2-carboxamide
3-methyl-7-[1-(pyridine-4-carbonyl)piperidin-4-yl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
5-cyclobutanecarbonyl-1'-(pyridine-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-{3-[2-(azocan-1-yl)-2-oxoethyl]morpholin-4-yl}-2-(pyridin-3-yl)ethan-1-one
4-chloro-3-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}-1-methyl-1H-indazole
1-tert-butyl-5-oxo-N-[2-(pyrazin-2-yl)ethyl]pyrrolidine-3-carboxamide
ethyl 1-(1,3-benzothiazol-2-yl)-5-({[1-(thiophen-2-yl)propyl]amino}methyl)-1H-pyrazole-4-carboxylate
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-2-(thiophen-3-yl)acetamide
(4aR,8aS)-N,N-dimethyl-1-(3,4,5-trifluorobenzoyl)-decahydro-1,6-naphthyridine-6-sulfonamide
1-[(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octan-8-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one