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[(3R,4R)-4-(morpholin-4-ylmethyl)-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]pyrrolidin-3-yl]methanol
5,6-dimethyl-N-[2-(1-methylpyrrolidin-2-yl)ethyl]pyridine-3-carboxamide
1-(propan-2-yl)-4-{1-[3-(1H-pyrazol-5-yl)phenyl]piperidin-4-yl}-1,4-diazepane
2-amino-4-[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-methyl-8-[2-(2-methyl-1H-indol-3-yl)acetyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[1-(5-chloropyridine-3-carbonyl)piperidin-2-yl]-5-fluoro-1H-1,3-benzodiazole
(1S,5R)-6-(2-methoxyethyl)-3-(3-methoxypyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-hydroxy-2-(4-methylphenyl)-N-[(3S)-piperidin-3-yl]pyrimidine-5-carboxamide
5,6-dichloro-2-(1,3-dimethyl-1H-pyrazol-5-yl)-1H-1,3-benzodiazole
(4aS,8aR)-6-(4-ethoxybenzoyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
3-methyl-1-(2-methylpropyl)-4-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]piperazin-2-one
6-(3-chlorophenyl)-7-(cyclopropylmethyl)-N-(2-hydroxybutyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-(carbamoylmethyl)-N-[1-(2,5-difluorophenyl)cyclopropyl]piperidine-3-carboxamide
1-{2-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]phenyl}ethan-1-one
5-[(dimethylamino)methyl]-N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}furan-2-carboxamide
(2R,4S)-4-hydroxy-1-[2-(3-methylphenyl)benzoyl]piperidine-2-carboxylic acid
2-(1-cyclohexyl-4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl)ethan-1-ol
1-{3-[({4-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)amino]propyl}pyrrolidin-2-one
2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]-N-methyl-N-(1,2-oxazol-3-ylmethyl)acetamide
1-[1-(2-oxobutanoyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-butyl-3-(3-methyl-1H-1,2,4-triazol-5-yl)-N-(3-phenylprop-2-yn-1-yl)propanamide
1-(4-methoxyphenyl)-4-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}piperazine
5-[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]pentan-1-ol
4-{[6-(4-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-3-methylpiperazin-2-one
1-[2-(8-methylquinolin-5-yl)pyrimidin-4-yl]piperidin-3-ol
1'-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)sulfonyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-cyclohexyl-3-(cyclopropylmethyl)-5-(thiomorpholine-4-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
4-{[3-oxo-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]amino}-1-phenylpyrrolidin-2-one
methyl 3-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(1R,2S)-2-{[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]amino}cyclopentane-1-carboxamide
N-{[3-(furan-2-ylmethoxy)-4-methoxyphenyl]methyl}-2,3-dimethyl-N-(oxolan-2-ylmethyl)-1H-indole-7-carboxamide
4-{5-[1-(benzenesulfonyl)cyclopropyl]-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl}-3-methylpyridine
N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-1H-1,2,3-benzotriazole-5-carboxamide
methyl 4-{[3-(5-fluoro-2-methoxybenzoyl)piperidine-1-carbonyl]amino}benzoate
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-(2-oxoazepan-3-yl)propanamide
(4aR,7aS)-1-(2-methoxyethyl)-4-(pent-2-yn-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-ethyl-6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-methoxy-1-{1'-[2-(piperidin-1-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
2-({[(3R,4R)-1-(1-benzofuran-5-ylmethyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-(1-butyl-1H-pyrazol-5-yl)-4-(4-methoxybenzoyl)piperazine-1-carboxamide
N-(1-{2-[4-(4-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-3-(2-methoxyphenyl)propanamide
2-methyl-3-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1H-indol-4-one
1-cyclopropanecarbonyl-N-methyl-N-[(4-phenoxyphenyl)methyl]pyrrolidine-2-carboxamide
(1S,5R)-6-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
7-(cyclobutylmethyl)-2-[2-(2-oxoazepan-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amine
N-[(3S,4R)-4-hydroxyoxolan-3-yl]-5-(2-methoxyphenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
3-ethyl-1-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}urea