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5-[(3,4-difluorophenyl)methyl]-4-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-{4-[3-(dimethylamino)propyl]piperazin-1-yl}-2-(2,4-dimethylphenyl)acetic acid
1-(thiophen-2-ylmethyl)-4-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperazine
1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-2-[3-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]ethan-1-one
5-ethyl-2-methyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]pyrimidin-4-amine
2-(3-chlorophenoxy)-1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl]methanol
6-methyl-N4-[1-(6-methylpyridin-2-yl)ethyl]-5-(prop-2-en-1-yl)pyrimidine-2,4-diamine
5-[(dimethylamino)methyl]-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-1,3,4-oxadiazole-2-carboxamide
1-methyl-4-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]piperazine-2-carboxylic acid
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(3-methylphenoxy)ethan-1-one
methyl[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl](quinoxalin-6-ylmethyl)amine
3-(5-methylfuran-2-yl)-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
4-[(2,3-difluorophenyl)methyl]-7-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-ethyl-6-[9-oxo-8-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-3-carboxamide
2,3,4-trimethoxy-N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
N,5,7-trimethyl-N-(oxan-4-ylmethyl)pyrido[2,3-d]pyrimidin-4-amine
N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-propylpyrrolidin-3-yl]-1-methyl-1H-pyrazole-3-carboxamide
1-{4-[4-(2-hydroxypropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-2-(2H-indazol-2-yl)ethan-1-one
6-({methyl[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)-1,4-oxazepan-6-ol
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-{[7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
7-(cyclohexylmethyl)-2-(1,3-thiazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-methyl-N-[2-methyl-5-(2-{[methyl(propan-2-yl)amino]methyl}propanamido)phenyl]benzamide
1-[(3-fluorophenyl)methyl]-6-oxo-N-(3-phenylpropyl)piperidine-3-carboxamide
1-{5-[3-(cyclopropylmethyl)-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-1H-pyrazol-3-yl}ethan-1-one
3,3-dimethyl-1-({5-[(2,3,4-trifluorophenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)urea
(3S,4R)-1-(2-ethylpyrimidine-5-carbonyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
8-[(4-hydroxyphenyl)methyl]-1-(2-methoxyethyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-3-yl)methanamine
1-(1,3-benzothiazol-2-yl)-N-[3-(pyridin-3-yl)propyl]piperidin-4-amine
(3R,4R)-1-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-4-(4-methylpiperazin-1-yl)piperidin-3-ol
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-1,2,3-triazole-5-carboxamide
N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]piperidine
3-(1-butyl-1H-imidazol-2-yl)-N-[4-(methylsulfanyl)phenyl]piperidine-1-carboxamide
6-methyl-2-({[2-(1-propylpiperidin-4-yl)ethyl]amino}methyl)quinolin-4-ol
3-(3-fluorophenyl)-N-[(3-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)propanamide
2-[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]-1H-1,3-benzodiazole-5-carboxylic acid
(3S,4R)-1-({2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidin-5-yl}methyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
2-cyclopentyl-9-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}-2,9-diazaspiro[5.5]undecan-3-one
N,3-dimethyl-N-[1-(pyridin-2-yl)propyl]furan-2-carboxamide
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
ethyl 5-(1,3-benzothiazol-2-ylmethyl)-1-[2-(dimethylamino)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-{[(1r,4r)-4-hydroxycyclohexyl]amino}pyridine-3-carboxamide
N-[(1S,2R)-2-aminocyclobutyl]-6-methyl-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-8-carboxamide
{2-[(6-methoxypyridin-2-yl)oxy]hex-5-en-1-yl}(methyl)(pyridin-3-ylmethyl)amine
N-[4-(5-methylfuran-2-amido)phenyl]piperidine-3-carboxamide
4-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetyl]-1-(2-methoxyphenyl)piperazin-2-one
(3S,4R)-4-(2-methoxyphenyl)-1-{2-[methyl(piperidin-4-yl)amino]acetyl}pyrrolidine-3-carboxylic acid