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N-[2-({[(2-fluorophenyl)methyl](2-methoxyethyl)amino}methyl)quinolin-6-yl]acetamide
N-[4-(3-fluorophenyl)phenyl]-1-methylpyrrolidine-2-carboxamide
4-{[4-(3-hydroxyprop-1-yn-1-yl)phenyl]methyl}-1-phenylpiperazin-2-one
N-[(3R,4R)-4-hydroxypyrrolidin-3-yl]-4-(4-oxo-3,4-dihydroquinazolin-3-yl)butanamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carboxamide
N-(1,4-dioxan-2-ylmethyl)-2,3-dihydro-1,4-benzodioxine-5-carboxamide
7-fluoro-2-methyl-N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}quinoline-4-carboxamide
[(3R,5R)-5-[(dimethylamino)methyl]-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]methanol
2-methyl-N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)propanamide
[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl][(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]methylamine
1-[(5-ethylfuran-2-yl)methyl]-3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
N,1-bis(propan-2-yl)-2-(pyridin-4-yl)-1H-1,3-benzodiazole-5-sulfonamide
1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-4-(2-methoxybenzoyl)piperazine
3-{methyl[2-(methylcarbamoyl)ethyl]sulfamoyl}-N-(pyrrolidin-3-yl)benzamide
2,6-dimethyl-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)quinoline-4-carboxamide
1-(4-chlorophenyl)-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}cyclobutane-1-carboxamide
1-methyl-4-[4-(2-phenoxyethyl)piperazine-1-carbonyl]imidazolidin-2-one
3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methyl-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]propanamide
5-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
2-(dimethylamino)-4-methyl-N-[(1-propyl-1H-imidazol-2-yl)methyl]pyrimidine-5-carboxamide
methyl (2S)-2-({1-[4-(2-phenoxyacetamido)phenyl]piperidin-4-yl}amino)-2-phenylacetate
N-tert-butyl-8-(2-methoxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
5-(diethylamino)-1-ethyl-N-(furan-2-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-ethyl-3-(1-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}piperidin-4-yl)-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2,2-dimethyl-N-(1-{1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
4-(3-methyl-3-phenylpiperidin-1-yl)pyrimidin-2-amine
8-[(2-cyclohexylpyrimidin-5-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
4-benzyl-3-cyclobutyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-(2-fluoro-5-methanesulfonamidophenyl)-3-(3-methyl-1,1-dioxo-1λ6-thiolan-3-yl)urea
N-ethyl-1-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]pyrrolidine-3-carboxamide
3-{[4-({2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}amino)-6-methylpyrimidin-2-yl]amino}phenol
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)cyclobutanecarboxamide
methyl({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)[1-(pyridin-2-yl)ethyl]amine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-3-(5-phenyl-1,3,4-oxadiazol-2-yl)propanamide
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(3S)-N,N-dimethyl-1-[2-methyl-7-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]pyrrolidin-3-amine
1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-4-(4-propyl-1H-1,2,3-triazol-1-yl)piperidine
1-(oxan-4-yl)-N-{[2-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
4-(2H-1,3-benzodioxol-5-yl)-2-{[(9H-fluoren-9-yl)amino]methyl}phenol
N-[4-({[2-(2-oxoimidazolidin-1-yl)ethyl]carbamoyl}methyl)phenyl]butanamide
3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-[(1-methyl-1H-indol-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(4-fluorophenyl)methyl]-4-(3-methyl-1H-pyrazole-4-carbonyl)morpholine
2-{methyl[5-({methyl[(1-methylpiperidin-3-yl)methyl]amino}methyl)pyrimidin-2-yl]amino}acetic acid
6-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-9H-purine
1-{2-[(3,5-dimethylphenyl)formamido]ethyl}-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-[(3S,4R)-1-(2-ethylpyridine-4-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
N-[(3S,4R)-1-[(1-benzyl-1H-imidazol-2-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
3-(2-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
5-methoxy-3-{[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]methyl}-1H-indazole
N-{3-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-3-oxopropyl}methanesulfonamide