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6-methyl-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-3-(thiomorpholine-4-carbonyl)-1,4-dihydropyridin-4-one
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-N'-(4-methylphenyl)propanediamide
5-[(cyclopropylmethyl)(propyl)amino]-1-methyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-{1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]piperidin-4-yl}pyridine
(2S)-3-hydroxy-2-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}propanamide
6-methyl-4-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydropyridin-2-one
(2r,4r)-2-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-5,7-diazaspiro[3.4]octane-6,8-dione
5-fluoro-2-[1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
1-(4-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}phenyl)imidazolidine-2,4-dione
4-methyl-5-{1-[(1-methylpiperidin-3-yl)methyl]-1H-pyrazol-3-yl}-N-[(2,4,5-trimethoxyphenyl)methyl]-1,3-thiazol-2-amine
5-fluoro-2-[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]-1H-1,3-benzodiazole
5-ethyl-N4-[2-methoxy-1-(pyridin-2-yl)ethyl]pyrimidine-2,4-diamine
4-(2-propyl-1,3-thiazole-4-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
[(4aS,8aR)-6-[(2-methyl-1,3-oxazol-4-yl)methyl]-decahydro-1,6-naphthyridin-4a-yl]methanol
4-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
6-[3-(3-methoxypropyl)piperidine-1-carbonyl]-2-methyl-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
N-[2-(1,4-dioxo-1,2,3,4-tetrahydrophthalazin-2-yl)ethyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
N4-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}pyrimidine-4,6-diamine
N-{4-[2-(1H-imidazol-1-yl)propanamido]phenyl}-5-methylfuran-3-carboxamide
4-(4-methoxyphenyl)-4-oxo-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]butanamide
4-(2-oxooxolan-3-yl)-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-3-one
4-methoxy-N-{[1-(pyridin-2-ylmethyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
2-(butylsulfanyl)-6-[3-(morpholine-4-carbonyl)piperidin-1-yl]pyrimidin-4-amine
1-(2-methoxyphenyl)-4-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}piperazin-2-one
2-[methyl({2-[2-(prop-2-en-1-yl)phenoxy]ethyl})amino]acetic acid
4-methyl-N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
2-(2-methoxyethyl)-9-[(2-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
N-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-4-(6-methylpyridin-2-yl)piperazine-1-carboxamide
6-methyl-2-({[3-(pyridin-4-yl)propyl]amino}methyl)quinolin-4-ol
methyl 4-({[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]carbamoyl}amino)-3-methylbenzoate
6-fluoro-2-{[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methyl}quinolin-4-ol
6-fluoro-2-oxo-N-(3-phenylprop-2-yn-1-yl)-N-(prop-2-en-1-yl)-1,2-dihydroquinoline-4-carboxamide
2-({4-[(3,4-difluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
2-(4-fluorophenyl)-1-(4-methanesulfonylbenzoyl)piperidine
1-{2-hydroxy-3-[4-({[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]amino}methyl)-2-methoxyphenoxy]propyl}piperidin-4-ol
N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}-3-azaspiro[5.5]undecan-9-amine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(morpholin-4-yl)propanamide
2-(3-hydroxypropyl)-9-(quinolin-6-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-({3-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]thiophene-2-carboxamide
4-(5-{[4-(dimethylsulfamoyl)piperazin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoic acid
1-{2-[2-(thiophen-2-yl)ethyl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
4-(4-methoxyphenoxy)-1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]piperidine
2-(adamantan-1-yl)-4-hydroxy-N-[2-(pyrrolidin-1-yl)propyl]pyrimidine-5-carboxamide
(3R,4R)-3-cyclopropyl-4-methyl-1-(pyridin-4-yl)pyrrolidin-3-ol
2-[3-(6-methoxypyridin-3-yl)-1H-indazol-1-yl]-N-(1-methyl-1H-1,2,3-triazol-4-yl)acetamide
1-[1-(4-{[2-(2-fluorophenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)piperidin-4-yl]piperidin-4-ol
2-amino-6-(4-fluoro-2-methylphenyl)-4-[5-(hydroxymethyl)furan-2-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
5-[(1-benzylpiperidin-4-yl)amino]-1-(cyclohexylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-(pyridin-2-yl)-N-{[1-(pyridin-2-yl)piperidin-3-yl]methyl}pyrimidin-2-amine