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8-[4-(benzyloxy)butyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(1S,3R)-3-[1-(4-chloro-2-methylphenyl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]cyclohexan-1-amine
2-[4-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)phenoxy]-1-(morpholin-4-yl)ethan-1-one
4-[3-(propan-2-yl)-1H-pyrazol-1-yl]-1-{thieno[2,3-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
N-[5-chloro-2-(1H-1,2,4-triazol-1-yl)phenyl]-3-(1H-imidazol-1-ylmethyl)piperidine-1-carboxamide
N-[3-(2-oxo-1,2-dihydropyridin-1-yl)propyl]-3-(pyridin-3-yl)propanamide
3-(5-fluoro-2-methoxybenzoyl)-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-ethyl-N-methyl-5-oxopyrrolidine-3-carboxamide
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3,4-difluorophenyl)acetamide
2-[(3R,4S)-3-[(morpholine-4-sulfonyl)amino]-4-propylpyrrolidin-1-yl]acetamide
N,4-dimethyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-3-(2-oxoimidazolidin-1-yl)benzamide
2-{1-cyclohexyl-4-[(8-methoxy-2H-chromen-3-yl)methyl]piperazin-2-yl}ethan-1-ol
[(5-{1-[(4-methoxy-3-methylphenyl)methyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
4-(3-{2-oxa-7-azaspiro[4.5]decane-7-carbonyl}phenyl)-1λ6-thiomorpholine-1,1-dione
4-(1H-imidazol-1-yl)-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]butanamide
N-[4-(propan-2-yl)phenyl]piperidin-3-amine
(2S,4R)-N-(2-methoxyethyl)-4-{[(4-phenylphenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
2-{[1-(2-ethoxypyridine-3-carbonyl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
1-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-N-(4-methylpentan-2-yl)piperidin-4-amine
6-[(1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]quinoline
2-{[(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
4,6-dimethyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
3-(5-{[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
2-(2-methylphenyl)-N-[(1-methylpiperidin-3-yl)methyl]benzamide
3-{1-[(2S)-2-amino-3-(1H-imidazol-4-yl)propanoyl]piperidin-4-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1'-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
3-{[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]methyl}pyridine
1-(2-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
N-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
(4aS,8aR)-1-(3-methylbutyl)-6-(1H-pyrazole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-[1-(4-methylpyrimidin-2-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
2-(4-methoxy-2-methylphenyl)-2-{methyl[2-(pyrrolidin-1-yl)ethyl]amino}acetic acid
N-[(3-tert-butyl-1,2,4-oxadiazol-5-yl)methyl]-4-(3-hydroxy-3-methylbutyl)benzamide
4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-N,N-dimethylpiperidine-1-carboxamide
2-{[4-(5-chloropyrimidin-2-yl)piperazin-1-yl]methyl}quinolin-8-ol
(4R)-N,3-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1,3-thiazolidine-4-carboxamide
3-(1,3-benzothiazol-2-yl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}propanamide
N-cyclopentyl-5-(2-ethylpiperidine-1-carbonyl)-1-[(3-methoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
N-(2-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)pyridine-4-carboxamide
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
2-(2,5-dioxoimidazolidin-4-yl)-N-({3-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)acetamide
(3S,4S)-4-cyclopropyl-1-[2-hydroxy-6-(trifluoromethyl)pyridine-3-carbonyl]pyrrolidine-3-carboxylic acid
N-tert-butyl-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
1-(furan-2-ylmethyl)-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]piperidine-3-carboxamide
[(5-{1-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-3-(methylsulfanyl)propan-1-one
1-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-4-amine