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2-[5-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
N-(2,3-dihydro-1H-inden-2-yl)-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
(2R,4S)-1-[2-(2-ethoxyethoxy)benzoyl]-4-hydroxypiperidine-2-carboxylic acid
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-N'-(4-methylphenyl)propanediamide
1-[5-(methoxymethyl)thiophene-2-carbonyl]-3-(3-methylphenoxy)azetidine
N-cyclopentyl-5-(4-hydroxy-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)-1-benzofuran-2-carboxamide
2-[4-({[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)phenyl]-3H,4H,5H,6H,7H-cyclopenta[d]pyrimidin-4-one
3-{[1-(2,6-dimethylhept-5-en-1-yl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
1-[3-(morpholin-4-yl)propyl]-6-oxo-N-[2-(pyridin-3-yloxy)ethyl]piperidine-3-carboxamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
5-{2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N,2,3,5-tetramethyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
5-(methoxymethyl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
5-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidine-1-carbonyl]pyridine-2-carbonitrile
2-amino-6-(2-amino-5-methyl-1,3-thiazol-4-yl)-4-(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-[2-(diethylamino)ethyl]-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-hydroxy-2-methyl-1-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]propan-1-one
2-({3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1,3-thiazole
7-methyl-3-{[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
(1R,5R)-6-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[4-(dimethylamino)azepan-1-yl]-2-(5-ethyl-1-benzofuran-3-yl)ethan-1-one
2-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[5-(2-cyclohexylethyl)-1,3,4-oxadiazol-2-yl]-N-[(4-methylphenyl)methyl]propanamide
(2S,4S)-4-amino-N,N-diethyl-1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]pyrrolidine-2-carboxamide
1-[1-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)piperidin-4-yl]piperidin-4-ol
1-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
3-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-1-(pyrrolidin-1-yl)propan-1-one
3-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)-1-[(4-hydroxyphenyl)methyl]urea
2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methylpyridine-3-carbonitrile
methyl 4-(5-{[methyl(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoate
1-cyclobutanecarbonyl-N-[(2,6-dimethylpyridin-4-yl)methyl]piperidine-4-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-2-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
6-(2-ethoxybenzoyl)-2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
2-(2-chloro-4-{[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]methyl}-6-methoxyphenoxy)acetic acid
2-oxo-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}-1,2-dihydroquinoline-4-carboxamide
4-(3-benzyl-1H-pyrazol-5-yl)-1-(1-ethyl-1H-pyrazole-5-carbonyl)piperidine
9-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[(dimethylamino)methyl]-N-ethyl-N-[2-(3-methylphenoxy)ethyl]-1,3-thiazole-4-carboxamide
4-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-N-methylpyridin-2-amine
2-{[(1R,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1H-1,3-benzodiazole
methyl({[1-(2-methylpropyl)-2-(oxolan-2-ylmethanesulfonyl)-1H-imidazol-5-yl]methyl})(pyridin-2-ylmethyl)amine
N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2-(pyridin-4-ylsulfanyl)acetamide
(3S,4R)-4-(hydroxymethyl)-1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-3-ol
N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
N,N,3-trimethyl-4-({[3-(oxolan-3-yl)propyl]carbamoyl}amino)benzamide
2-[2-methyl-4-oxo-1-(oxolan-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]-N-(thiophen-3-ylmethyl)acetamide
1-[3-cyclopentyl-5-(1H-indazol-3-yl)-1H-1,2,4-triazol-1-yl]butan-2-ol
(2R,6R)-4-[(dimethyl-1,3-thiazol-5-yl)methyl]-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-methoxy-5-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]pyridine