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N-[(4-methanesulfonylmorpholin-2-yl)methyl]-5-phenyl-1H-pyrazole-3-carboxamide
1-{2-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-[1-(thiophen-2-yl)propyl]piperidine-4-carboxamide
N-[(3,5-dimethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
3-[2-(dimethylamino)ethyl]-5-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
1-[4-(morpholine-4-carbonyl)phenyl]-N-[1-(1,3-thiazol-2-yl)ethyl]piperidin-4-amine
3-[3-(2-{[(2-chlorophenyl)methyl]carbamoyl}ethyl)piperidine-1-carbonyl]pyridin-1-ium-1-olate
1-{2,8-diazaspiro[4.5]decane-3-carbonyl}-4-(4-fluorophenyl)piperidin-4-ol
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-2-(ethylamino)-N-methylpyrimidine-5-carboxamide
N-[(2R,3R)-1'-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-(2,2-difluoroethyl)-6-(2,5-dimethylfuran-3-yl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-ethyl-N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1H-indole-5-carboxamide
N-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
5-{[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-N,N-dimethylpyridin-2-amine
N-(2-methoxyethyl)-3-(3-methoxyphenyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-4-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-3-phenylpropanamide
N-{1-[1-(1H-indole-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
1-[3-(2-phenylpropyl)-1,2-oxazole-5-carbonyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
4-methoxy-N-(2-methoxyethyl)-2-[(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)oxy]benzamide
N-[2-(5-methylthiophen-2-yl)ethyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-{3,9-diazaspiro[5.6]dodecan-9-yl}-3-(3,5-dimethyl-1H-pyrazol-4-yl)propan-1-one
2-(1H-1,3-benzodiazol-1-ylmethyl)-N-[(5-methylpyrazin-2-yl)methyl]-1,3-oxazole-4-carboxamide
1-phenyl-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-1,2,3-triazole-4-carboxamide
1-{4-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
4-[4-({3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)phenyl]but-3-yn-1-ol
6-(2,5-dimethylfuran-3-yl)-N,7-dimethyl-8-oxo-N-pentyl-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-[(dimethylamino)methyl]-4-{1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-2-yl}phenol
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-3-[3-(2-oxopyrrolidin-1-yl)propyl]urea
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(2-methoxy-4-methylbenzoyl)pyrrolidin-3-yl]methanol
8-chloro-2-[1-(pyridin-3-yl)-1H-imidazol-2-yl]quinoline
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}butanamide
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]benzamide
methyl 7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-3-(3-phenylpropanoyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-2-(4-methyl-1,4-diazepan-1-yl)acetamide
4-[4-(cyclohexylmethyl)-1H-1,2,3-triazol-1-yl]-1-[(2R)-pyrrolidin-2-ylmethyl]piperidine
N-[2-(2-fluorophenoxy)ethyl]-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
N-(2-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}ethyl)-3-methylthiophene-2-carboxamide
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}acetamide
2-[2-(1-{2-[4-(hydroxymethyl)phenyl]acetyl}piperidin-3-yl)-1H-imidazol-1-yl]acetamide
2-(4-fluorophenyl)-1-[1-(methoxymethyl)cyclobutanecarbonyl]azetidine
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methylpiperidine
N-[(1R,3R)-3-aminocyclopentyl]-2,3-dichlorobenzene-1-sulfonamide
N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propanamide
N-cyclopentyl-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(4-methylphenyl)(pyridin-4-yl)methyl]-4-(piperidin-1-yl)butanamide
N-[1-(pyridin-3-yl)pentyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
ethyl 2-{1-[1-(4-methylquinazolin-2-yl)piperidine-4-carbonyl]piperidin-2-yl}acetate
2-{2-[2-(6-methylpyridin-2-yl)-1H-imidazol-1-yl]ethyl}-1,2,3,4-tetrahydrophthalazine-1,4-dione
1-(oxolan-2-ylmethyl)-4-phenyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one