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2-methyl-5-{[(1R,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
methyl 5-(1,4-dioxane-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(2-oxo-1,2-dihydropyridin-1-yl)propanamide
1-(cyclohexylmethyl)-N,N-dimethyl-5-{[(3-methyl-1,2-oxazol-5-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-[2-oxo-4-(2-phenylbenzoyl)piperazin-1-yl]benzonitrile
N-ethyl-2-(1-ethyl-1H-pyrazol-4-yl)-5,7-dimethyl-N-(propan-2-yl)quinoline-4-carboxamide
2-[4-({[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}methyl)phenoxy]ethan-1-ol
(3R,4R)-4-{methyl[2-(pyridin-2-yl)ethyl]amino}-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-3-ol
1-{2-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridin-6-yl]-2-oxoethyl}-1,2,3,4-tetrahydroquinolin-2-one
1-(azepan-1-yl)-3-{3-[({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amino)methyl]phenoxy}propan-2-ol
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-1-oxo-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
methyl 4-({2-[(4-methoxyphenyl)methyl]morpholin-4-yl}methyl)benzoate
2-{2-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}pyridine
1-methyl-5-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-3-propyl-1H-pyrazole
2-[3-(3-methoxyphenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[(3-methylpyridin-2-yl)methyl]acetamide
3-{3-[5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]propyl}pyridine
2-amino-N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
9-(5,6-dimethylpyridine-3-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-4-(pyridin-3-ylmethyl)piperazine
[(3R,4S)-4-[(4-methylpiperazin-1-yl)methyl]-1-(2-phenylethyl)pyrrolidin-3-yl]methanol
4-{3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl}-2-methylphenol
N,N-diethyl-2-(2-ethylpyrimidin-5-yl)-3,6-dimethylquinoline-4-carboxamide
1-{1-[2-(1H-indazol-3-yl)acetyl]piperidin-4-yl}-N-(propan-2-yl)piperidine-4-carboxamide
(3S,4S)-4-cyclopropyl-1-({[2-(4-fluorophenyl)ethyl]carbamoyl}methyl)pyrrolidine-3-carboxylic acid
N-[(2-aminopyridin-3-yl)methyl]-4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
N-{[1-(2H-1,3-benzodioxol-5-yl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]methyl}benzamide
(2S)-2-{5-[4-ethoxy-3-(hydroxymethyl)phenyl]-4-phenyl-1H-imidazol-1-yl}-3-methylbutanamide
1-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-4-(6-methylpyridin-2-yl)piperazine
1-[(2-methoxyphenyl)methyl]-6-oxo-N-[3-(pyridin-2-yl)propyl]piperidine-3-carboxamide
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-2-(methylamino)-1,3-thiazole-4-carboxamide
1-(2-methoxyacetyl)-N-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxamide
6-fluoro-2-(1-methyl-1H-pyrazol-4-yl)-4-{octahydro-1H-pyrido[1,2-a]piperazine-2-carbonyl}quinoline
N-(2-methylpropyl)-1-[1-(1-propylpiperidin-4-yl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
2-(2H-1,2,3-benzotriazol-2-yl)-N-{[2-(diethylamino)pyridin-3-yl]methyl}acetamide
methyl (2S,4S)-1-[(3-chlorophenyl)methyl]-4-[4-(1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
4-hydroxy-N-[(2S)-1-hydroxy-4-methylpentan-2-yl]-2-(4-methylphenyl)pyrimidine-5-carboxamide
1-[2-(3-benzyl-1H-1,2,4-triazol-5-yl)ethyl]-1H-1,3-benzodiazole
1-[(4-chlorophenyl)methyl]-N-[2-(5-methylfuran-2-yl)ethyl]-6-oxopiperidine-3-carboxamide
N-cyclopropyl-1-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-3-(2-oxopiperidin-1-yl)propanamide
1-[(4-fluorophenyl)methyl]-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
N-[(3-hydroxypyrrolidin-3-yl)methyl]naphthalene-1-carboxamide
N-[(7-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]thiophene-3-sulfonamide
benzyl 5-oxo-1,4,9-triazaspiro[5.5]undecane-9-carboxylate
1-(2-methylphenyl)-4-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]piperazin-2-one
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(4-methylpyrimidine-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-[({[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)methyl]-N-methylpyrimidin-2-amine
3-[1-(2,6-dimethoxypyrimidin-4-yl)piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(2-hydroxyethyl)-N-methylacetamide