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3-(2,3-dihydro-1H-inden-2-yl)-8-{[2-(furan-2-yl)phenyl]methyl}-1-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-(3-methoxyphenyl)-N-(oxolan-2-ylmethyl)acetamide
N-[2-(N-methylmethanesulfonamido)ethyl]-4-(piperidin-1-ylmethyl)benzamide
N-(4-fluoro-2-methylphenyl)-3-(1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidin-3-yl)propanamide
3-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(2-chlorophenyl)methyl]-3-(1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)propanamide
6-(3,4-dimethylpiperazin-1-yl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
7-chloro-4-methyl-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]quinolin-2-amine
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-2-(pyridin-4-yl)acetamide
ethyl 1-{5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperidine-3-carboxylate
N,N-bis(pyridin-3-ylmethyl)-2-(4H-1,2,4-triazol-4-yl)benzamide
3,5-dimethyl-1-{1-[(1-phenyl-1H-pyrazol-5-yl)methyl]pyrrolidin-3-yl}-1H-pyrazole
1-[2-(morpholin-4-yl)ethyl]-3-[3-(1H-1,2,4-triazol-1-yl)phenyl]urea
2-{4-[3-(ethanesulfonyl)phenyl]phenyl}-5-methyl-1,3,4-oxadiazole
5-[({[3-(2-{4-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperazin-1-yl}ethoxy)phenyl]methyl}(methyl)amino)methyl]pyrrolidin-2-one
(1S,9aR)-1-{[4-(3-methylphenyl)piperazin-1-yl]methyl}-octahydro-1H-quinolizine
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-3-methylpiperidine
7-(2-cyclohexylethyl)-2-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
2-(2-phenyl-1H-imidazol-1-yl)-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
(1S,5R)-6-[3-(4-methylphenyl)-1H-pyrazole-5-carbonyl]-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
(1S,5R)-N-[3-(1H-imidazol-5-yl)phenyl]-10-oxo-3,9-diazabicyclo[3.3.2]decane-3-carboxamide
2-{1-[(4-fluorophenyl)methyl]-4-(quinolin-2-ylmethyl)piperazin-2-yl}ethan-1-ol
4-[5-methyl-4-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)-2-oxopiperazin-1-yl]benzonitrile
1-{2-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
(1H-1,3-benzodiazol-2-ylmethyl)({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
N-[(3,4-dimethoxyphenyl)methyl]-2-{[(furan-2-ylmethyl)(prop-2-yn-1-yl)amino]methyl}-N-methylquinazolin-4-amine
N-[(2-methoxyphenyl)methyl]-N-(pyridin-4-ylmethyl)spiro[2.2]pentane-1-carboxamide
N-[3-(methylsulfanyl)propyl]-3-{[(3S)-piperidin-3-yl]sulfamoyl}benzamide
1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
N-butyl-N-methyl-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
(2R,6S)-2,6-dimethyl-4-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}morpholine
[(4-fluorophenyl)methyl]({[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl})(pyridin-4-ylmethyl)amine
1-{1'-[2-(4-fluorophenyl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(ethyl)(pyridin-4-ylmethyl)amine
N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
1-benzyl-4-[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-3-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N'-(3,5-dimethylphenyl)-N-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]propanediamide
4-(2-{[4-(4-methylphenyl)-5-(pyrimidin-5-yl)pyrimidin-2-yl]amino}ethyl)phenol
N3-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)piperidine-1,3-dicarboxamide
2-[(3S,4R)-3-cyclopropyl-4-[2-(2-ethoxyphenyl)acetamido]pyrrolidin-1-yl]acetic acid
methyl 5-[(4-hydroxybutan-2-yl)amino]-1-[2-(1H-indol-3-yl)ethyl]-3-(3-methoxypropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-(methoxymethyl)-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}cyclobutane-1-carboxamide
9-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
benzyl 3-{[(1,3-dimethyl-1H-pyrazol-4-yl)formamido]methyl}piperidine-1-carboxylate
N-{[2-(dimethylamino)-7-methylquinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]-3-(2-oxoimidazolidin-1-yl)benzamide
4-{2-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]-2-oxoethyl}-3,4-dihydro-2H-1,4-benzothiazin-3-one
5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-N-[2-(3-methylpyridin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
N4-methyl-N4-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
9-(2,4-difluorophenyl)-N-(2-methoxyethyl)-N,15-dimethyl-13-oxo-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide