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{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}({[3-(trifluoromethyl)phenyl]methyl})amine
N-cyclopropyl-3-[5-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
N-(2-{3-[(1R,5S)-6-azabicyclo[3.2.1]octane-6-carbonyl]benzenesulfonamido}ethyl)acetamide
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
2-[4-(4-benzylpiperazin-1-yl)piperidine-1-carbonyl]morpholine
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-1,2-dihydrophthalazin-1-one
3-[2-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-4-(furan-3-ylmethyl)piperazin-2-one
1-ethyl-5-(4-phenyl-1H-imidazol-5-yl)-1H-1,2,4-triazole
2-ethoxy-6-{[3-(2-hydroxyethyl)-4-(thiophen-3-ylmethyl)piperazin-1-yl]methyl}phenol
N,3,5,7-tetramethyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-1H-indole-2-carboxamide
4-amino-2-[4-(4-methyl-2,5-dioxoimidazolidin-4-yl)piperidin-1-yl]pyrimidine-5-carbonitrile
1-(cyclohexylmethyl)-N-methyl-N-[(3-methylpyridin-4-yl)methyl]-6-oxopiperidine-3-carboxamide
(3S,4S)-1-(2,2-dimethylpent-4-en-1-yl)-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
1-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-2-(2,4-dimethoxyphenyl)ethan-1-one
3-{imidazo[1,2-a]pyridin-2-ylmethyl}-6,7-dimethoxy-3,4-dihydroquinazolin-4-one
methyl 3-{[2-(1H-1,3-benzodiazol-1-yl)acetamido]methyl}-5-(4-fluorobenzenesulfonamido)benzoate
(1S)-1-[1-(2-methoxyphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-2-phenylethan-1-ol
6-(2-chlorophenyl)-2-{3-[(2-methylpyrrolidin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
4-({3-[6-(trifluoromethyl)pyridin-3-yl]phenyl}methyl)morpholine
4-(1-{[(2-methylpropyl)carbamoyl]methyl}piperidin-3-yl)benzoic acid
1-methyl-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-[(1-methyl-1H-indol-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2-methylphenyl)-4-{1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidin-3-yl}piperazine
3-[(2-fluorophenyl)formamido]-N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)propanamide
4-cyclobutyl-N-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]-6-methylpyrimidin-2-amine
N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-3-(1-methylpiperidin-2-yl)propanamide
2-{6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}-5-methyl-1H-1,3-benzodiazole
2-chloro-5-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-methylbenzamide
4-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]thiomorpholine
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
ethyl 4-{1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-yl}piperazine-1-carboxylate
2-(2-{1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
N-(2-hydroxypropyl)-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
3-[1-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]-1-(morpholin-4-yl)propan-1-one
3-{1-[(5-methylthiophen-2-yl)methyl]azetidin-3-yl}pyridine
3-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]butanamide
3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-[(2-methylphenyl)methyl]piperidine
1-(2-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}-2-oxoethyl)pyrrolidin-2-one
(1H-1,3-benzodiazol-2-ylmethyl)[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]methylamine
1-{6-[2-(trifluoromethyl)phenyl]pyridin-2-yl}ethan-1-ol
9-(butane-1-sulfonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
(1-phenoxypropan-2-yl)[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
6-methyl-2-{methyl[(1-phenylpyrrolidin-3-yl)methyl]amino}pyridine-3-carboxylic acid
3-(furan-2-yl)-3-[(3-methyl-1-propyl-1H-pyrazol-4-yl)formamido]propanoic acid
4-hydroxy-N-(2-phenoxyethyl)-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-(4-fluoro-2-methylphenyl)-3-{1-[2-(thiophen-3-yl)acetyl]piperidin-3-yl}propanamide