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3-(1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)-1-(pyrrolidin-1-yl)propan-1-one
N-[2-(1H-imidazol-1-yl)ethyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
8-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N,N-dimethyl-5-{[4-(quinazolin-4-yl)piperazin-1-yl]methyl}pyridin-2-amine
1-(pyridin-4-ylmethyl)-4-[4-(thiophen-3-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
N-(1-{1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]acetamide
(1S,5R)-6-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(2-hydroxyethyl)-9-[3-(pyridin-2-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(3-methyl-1-benzofuran-2-yl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
N-(pyrazin-2-yl)-2-{[2-(pyridin-3-yloxy)propyl]amino}acetamide
3-(3-methyl-1,1-dioxo-1λ6-thiolan-3-yl)-1-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
1-[2-(thiophen-2-yl)ethyl]-5-[2-({[3-(trifluoromethyl)phenyl]methyl}amino)ethyl]pyrrolidin-2-one
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,2-oxazole-3-carboxamide
2-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]pyrrolidin-2-yl}pyridine
2-(2,4-difluorophenoxy)-N-[2-(N-methylmethanesulfonamido)ethyl]acetamide
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(1H-imidazol-1-yl)ethan-1-one
1-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}azetidin-3-amine
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-[2-(6-methylpyridin-2-yl)ethyl]acetamide
1-(2H-1,3-benzodioxole-5-carbonyl)-4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidine
2-methyl-N-[2-(1H-pyrazol-3-yl)pyridin-3-yl]propanamide
N-ethyl-6-(2-fluorophenyl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-methyl-N-{2-[(pyridin-3-yl)amino]ethyl}-1,3-benzothiazole-6-carboxamide
1-cyclohexyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-4-oxo-5-(pyrrolidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
(2S,4R)-4-(2,3,6-trimethylquinoline-4-amido)pyrrolidine-2-carboxylic acid
N-[(3S)-2-oxoazepan-3-yl]-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-1,3-thiazole-5-carboxamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-4-methoxypiperidine-1-sulfonamide
N-cyclopropyl-3-(dimethyl-1,2-oxazol-4-yl)-N-(thiophen-3-ylmethyl)propanamide
{2-[({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)(isoquinolin-5-ylmethyl)amino]ethyl}dimethylamine
2,3,5,6-tetramethyl-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)benzamide
1-(4-hydroxypiperidin-1-yl)-3-[5-(pyridin-4-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propan-1-one
methyl 6-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-3-(furan-3-amido)thieno[2,3-b]pyridine-2-carboxylate
3-(azepane-1-carbonyl)-1-(prop-2-en-1-yl)-N-(pyridin-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[1-benzoyl-4-(pyrrolidin-1-ylmethyl)piperidin-4-yl]-5-methylpyridine
4-{[2-(cyclopropylmethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]methyl}benzoic acid
1-methyl-1-[2-(4-methylphenoxy)ethyl]-3-[2-(oxolan-2-ylmethoxy)phenyl]urea
N-[1-(2-methoxyphenyl)propan-2-yl]-N,2-dimethyl-4-phenylpyrimidine-5-carboxamide
N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]cyclohexanecarboxamide
N-cyclopropyl-2-[4-(2-phenylphenyl)-1H-1,2,3-triazol-1-yl]acetamide
N-[2-(2-chlorophenyl)-1-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]ethyl]-N-methylfuran-2-carboxamide
(1R,5R)-6-(2-fluorobenzoyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N2-[(4-methylphenyl)methyl]-N2-(2-methylpropyl)pyrrolidine-1,2-dicarboxamide
3-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1-(5-methanesulfonamido-2-methylphenyl)urea
2-methoxy-1-{1'-[5-(methoxymethyl)furan-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
3-[1-(4-aminopyrimidin-2-yl)piperidin-4-yl]-4-benzyl-4,5-dihydro-1H-1,2,4-triazol-5-one
5-chloro-N-[3-(1H-indazol-1-yl)propyl]-2,3-dihydro-1H-indole-2-carboxamide
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(2-methoxyethyl)methylamine
6-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
4-(2-methyl-1H-imidazol-1-yl)-1-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]piperidine-4-carboxylic acid
6-ethyl-N-[2-(1H-imidazol-4-yl)ethyl]-4-methylquinolin-2-amine